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TargetNorepinephrine transporter
LigandBDBM50003571
Substrate/Competitorn/a
Ki 340±n/a nM
CommentsPDSP_646
Citation Codd EEShank RPSchupsky JJRaffa RB Serotonin and norepinephrine uptake inhibiting activity of centrally acting analgesics: structural determinants and role in antinociception. J Pharmacol Exp Ther 274:1263-70 (1995) [PubMed]
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Norepinephrine transporter
Name:Norepinephrine transporter
Synonyms:n/a
Type:Enzyme Catalytic Domain
Mol. Mass.:2082.45
Organism:RAT
Description:Norepinephrine transporter 0 RAT::Q9JIA2
Residue:19
Sequence:
MLLARMKPQVQPELGGADQ
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BDBM50003571
n/a
NameBDBM50003571
Synonyms:(-)-3-Hydroxy-N-methylmorphinan hydrochloride (levorphanol) | 17-methyl-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-trien-4-ol | 17-methyl-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-trien-4-ol | Dextrorphan | Levorphanol
TypeSmall organic molecule
Emp. Form.C17H23NO
Mol. Mass.257.3706
SMILESCN1CCC23CCCCC2C1Cc1ccc(O)cc31 |TLB:0:1:9:18.12.11,THB:17:18:9:1.3.2|
Structure
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