Reaction Details |
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Target | Neuropeptide Y receptor type 1 |
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Ligand | BDBM50015490 |
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Substrate/Competitor | n/a |
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Ki | 0.09±n/a nM |
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Comments | PDSP_1377 |
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Citation | Bard, JA; Walker, MW; Branchek, TA; Weinshank, RL Cloning and functional expression of a human Y4 subtype receptor for pancreatic polypeptide, neuropeptide Y, and peptide YY. J Biol Chem270:26762-5 (1995) [PubMed] Article |
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More Info.: | Get all data from this article |
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Neuropeptide Y receptor type 1 |
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Name: | Neuropeptide Y receptor type 1 |
Synonyms: | NPY-Y1 | NPY1-R | NPY1R | NPY1R_HUMAN | NPYR | NPYY1 | neuropeptide Y receptor Y1 |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 44399.07 |
Organism: | Homo sapiens (Human) |
Description: | NPY-Y1 NPY1R HUMAN::P25929 |
Residue: | 384 |
Sequence: | MNSTLFSQVENHSVHSNFSEKNAQLLAFENDDCHLPLAMIFTLALAYGAVIILGVSGNLA
LIIIILKQKEMRNVTNILIVNLSFSDLLVAIMCLPFTFVYTLMDHWVFGEAMCKLNPFVQ
CVSITVSIFSLVLIAVERHQLIINPRGWRPNNRHAYVGIAVIWVLAVASSLPFLIYQVMT
DEPFQNVTLDAYKDKYVCFDQFPSDSHRLSYTTLLLVLQYFGPLCFIFICYFKIYIRLKR
RNNMMDKMRDNKYRSSETKRINIMLLSIVVAFAVCWLPLTIFNTVFDWNHQIIATCNHNL
LFLLCHLTAMISTCVNPIFYGFLNKNFQRDLQFFFNFCDFRSRDDDYETIAMSTMHTDVS
KTSLKQASPVAFKKINNNDDNEKI
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BDBM50015490 |
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n/a |
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Name | BDBM50015490 |
Synonyms: | CHEMBL438945 | H-YPSKPDNPGEDAPAEDMARYYSALRHYINLITRQRY-NH2 | NPY | NPY, human | NPY, human, rat | Tyr-Pro-Ser-Lys-Pro-Asp-Asn-Pro-Gly-Glu-Asp-Ala-Pro- Ala-Glu-Asp-Met-Ala-Arg-Tyr-Tyr-Ser-Ala-Leu-Arg-His- Tyr-Ile-Asn-Leu-Ile-Thr-Arg-Gln-Arg-Tyr-NH2 (NPY) | human Neuropeptide Y |
Type | Small organic molecule |
Emp. Form. | C189H285N55O57S |
Mol. Mass. | 4271.685 |
SMILES | n/a |
Structure |
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