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Target5-hydroxytryptamine receptor 7
LigandBDBM35256
Substrate/Competitorn/a
Ki 107.15±n/a nM
CommentsPDSP_1235
Citation To, ZPBonhaus, DWEglen, RMJakeman, LB Characterization and distribution of putative 5-ht7 receptors in guinea-pig brain. Br J Pharmacol115:107-16 (1995) [PubMed]  Article
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5-hydroxytryptamine receptor 7
Name:5-hydroxytryptamine receptor 7
Synonyms:5-HT7 | 5-HT7L | 5HT7R_CAVPO | HTR7 | Serotonin 7 (5-HT7) receptor
Type:Enzyme Catalytic Domain
Mol. Mass.:49632.36
Organism:GUINEA PIG
Description:5-HT7 HTR7 GUINEA PIG::P50407
Residue:446
Sequence:
MMGVNSSGRPDLYGHLHSILLPGRGLPDWSPDGGADPGVSTWTPRLLSGVPEVAASPSPS
WDGTWDNVSGCGEQINYGRAEKVVIGSILTLITLLTIAGNCLVVISVCFVKKLRQPSNYL
IVSLALADLSVAVAVIPFVSVTDLIGGKWIFGHFFCNVFIAMDVMCCTASIMTLCVISID
RYLGITRPLTYPVRQNGKCMPKMILSVWLLSASITLPPLFGWAQNVNDDKVCLISQDFGY
TIYSTAVAFYIPMSVMLFMYYRIYKAARKSAAKHKFPGFPRVQPESIISLNGMVKLQKEV
EECANLSRLLKHERKNISIFKREQKAATTLGIIVGAFTVCWLPFFLLSTARPFICGTACS
CIPLWVERTCLWLGYANSLINPFIYAFFNRDLRTTYRSLLQCQYRNINRKLSAAGMHEAL
KLAERPERPECVLQNSDYCRKKGHDS
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BDBM35256
n/a
NameBDBM35256
Synonyms:(S)-mianserin | Lerivon | MIANSERIN | MIANSERIN (+) | MIANSERIN (-) | Tolvon
TypeSmall organic molecule
Emp. Form.C18H20N2
Mol. Mass.264.3648
SMILES[H][C@]12CN(C)CCN1c1ccccc1Cc1ccccc21 |r|
Structure
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