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TargetGABA(A) receptor-associated protein
LigandBDBM50060321
Substrate/Competitorn/a
Ki>10000±n/a nM
CommentsPDSP_20
Citation Evans, BEBock, MGRittle, KEDiPardo, RMWhitter, WLVeber, DFAnderson, PSFreidinger, RM Design of potent, orally effective, nonpeptidal antagonists of the peptide hormone cholecystokinin. Proc Natl Acad Sci U S A83:4918-22 (1986) [PubMed]  Article
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GABA(A) receptor-associated protein
Name:GABA(A) receptor-associated protein
Synonyms:GABA A Benzodiazepine | GABA-A receptor subunit alpha 1
Type:Enzyme Catalytic Domain
Mol. Mass.:13921.89
Organism:GUINEA PIG
Description:D7RA28
Residue:117
Sequence:
MKFVYKEEHPFEKRRSEGEKIRKKYPDRVPVIVEKAPKARIGDLDKKKYLVPSDLTVGQF
YFLIRKRIHLRAEDALFFFVNNVIPPTSATMGQLYQEHHEEDFFLYIAYSDESVYGL
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  Blast E-value cutoff:
BDBM50060321
n/a
NameBDBM50060321
Synonyms:1H-Indole-2-carboxylic acid ((R)-1-methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-amide | 1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-amide | CCK antagonist synthetic 19 | CHEMBL419764
TypeSmall organic molecule
Emp. Form.C25H20N4O2
Mol. Mass.408.4519
SMILESCN1c2ccccc2C(=N[C@@H](NC(=O)c2cc3ccccc3[nH]2)C1=O)c1ccccc1 |c:9|
Structure
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