| Reaction Details |
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 | Report a problem with these data |
| Target | Cholecystokinin |
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| Ligand | BDBM21147 |
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| Substrate/Competitor | n/a |
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| Ki | 0.43±n/a nM |
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| Comments | PDSP_2196 |
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| Citation |  Pendley, CE; Fitzpatrick, LR; Capolino, AJ; Davis, MA; Esterline, NJ; Jakubowska, A; Bertrand, P; Guyon, C; Dubroeucq, MC; Martin, GE RP 73870, a gastrin/cholecystokinin-B receptor antagonist with potent anti-ulcer activity in the rat. J Pharmacol Exp Ther273:1015-22 (1995) [PubMed] |
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| More Info.: | Get all data from this article |
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| Cholecystokinin |
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| Name: | Cholecystokinin |
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| Synonyms: | CCK | CCKN_PIG | Cholecystokinin B |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 12528.64 |
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| Organism: | GUINEA PIG |
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| Description: | Cholecystokinin B 0 GUINEA PIG::P01356 |
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| Residue: | 114 |
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| Sequence: | MNGGLCLCVLMAVLAAGTLAQPVPPADSAVPGAQEEEAHRRQLRAVQKVDGESRAHLGAL
LARYIQQARKAPSGRVSMIKNLQSLDPSHRISDRDYMGWMDFGRRSAEEYEYTS
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| BDBM21147 |
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| n/a |
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| Name | BDBM21147 |
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| Synonyms: | (3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-amino-3-formamidopropanoic acid]-3-[4-(sulfooxy)phenyl]propanamido]-4-(methylsulfanyl)butanamido]acetamido}-3-(1H-indol-3-yl)propanamido]-4-(methylsulfanyl)butanamido]-3-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}propanoic acid | CCK-8 | CCK-8(SO3) | CHEMBL1121 | H-Asp-Tyr(SO3H)-Met-Gly-Trp-Met-Asp-Phe-NH2 | SINCALIDE | Syncalide | [125I]CCK-8 |
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| Type | radiolabeled ligand |
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| Emp. Form. | C49H62N10O16S3 |
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| Mol. Mass. | 1143.269 |
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| SMILES | CSCC[C@H](NC(=O)[C@H](Cc1ccc(OS(O)(=O)=O)cc1)NC(=O)[C@@H](N)CC(O)=O)C(=O)NCC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](Cc1ccccc1)C(N)=O |
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| Structure | 
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