| Reaction Details |
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 | Report a problem with these data |
| Target | Cholecystokinin |
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| Ligand | BDBM50061220 |
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| Substrate/Competitor | n/a |
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| Ki | 7.2±n/a nM |
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| Comments | PDSP_2199 |
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| Citation |  Pendley, CE; Fitzpatrick, LR; Capolino, AJ; Davis, MA; Esterline, NJ; Jakubowska, A; Bertrand, P; Guyon, C; Dubroeucq, MC; Martin, GE RP 73870, a gastrin/cholecystokinin-B receptor antagonist with potent anti-ulcer activity in the rat. J Pharmacol Exp Ther273:1015-22 (1995) [PubMed] |
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| More Info.: | Get all data from this article |
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| |
| Cholecystokinin |
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| Name: | Cholecystokinin |
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| Synonyms: | CCK | CCKN_PIG | Cholecystokinin B |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 12528.64 |
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| Organism: | GUINEA PIG |
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| Description: | Cholecystokinin B 0 GUINEA PIG::P01356 |
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| Residue: | 114 |
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| Sequence: | MNGGLCLCVLMAVLAAGTLAQPVPPADSAVPGAQEEEAHRRQLRAVQKVDGESRAHLGAL
LARYIQQARKAPSGRVSMIKNLQSLDPSHRISDRDYMGWMDFGRRSAEEYEYTS
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| BDBM50061220 |
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| n/a |
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| Name | BDBM50061220 |
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| Synonyms: | 1-((S)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-m-tolyl-urea | 1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-m-tolyl-urea | 1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-m-tolyl-urea((S)L365_260) | CHEMBL70380 | L-365,260 |
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| Type | Small organic molecule |
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| Emp. Form. | C24H22N4O2 |
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| Mol. Mass. | 398.4571 |
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| SMILES | CN1c2ccccc2C(=N[C@H](NC(=O)Nc2cccc(C)c2)C1=O)c1ccccc1 |c:9| |
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| Structure | 
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