| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Cholecystokinin |
|---|
| Ligand | BDBM82404 |
|---|
| Substrate/Competitor | n/a |
|---|
| Ki | 0.8±n/a nM |
|---|
| Comments | PDSP_2242 |
|---|
| Citation |  Pendley, CE; Fitzpatrick, LR; Capolino, AJ; Davis, MA; Esterline, NJ; Jakubowska, A; Bertrand, P; Guyon, C; Dubroeucq, MC; Martin, GE RP 73870, a gastrin/cholecystokinin-B receptor antagonist with potent anti-ulcer activity in the rat. J Pharmacol Exp Ther273:1015-22 (1995) [PubMed] |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| Cholecystokinin |
|---|
| Name: | Cholecystokinin |
|---|
| Synonyms: | CCK | CCKN_PIG | Cholecystokinin B |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 12528.64 |
|---|
| Organism: | GUINEA PIG |
|---|
| Description: | Cholecystokinin B 0 GUINEA PIG::P01356 |
|---|
| Residue: | 114 |
|---|
| Sequence: | MNGGLCLCVLMAVLAAGTLAQPVPPADSAVPGAQEEEAHRRQLRAVQKVDGESRAHLGAL
LARYIQQARKAPSGRVSMIKNLQSLDPSHRISDRDYMGWMDFGRRSAEEYEYTS
|
|
|
|---|
| BDBM82404 |
|---|
| n/a |
|---|
| Name | BDBM82404 |
|---|
| Synonyms: | Glycinamide,N-[[[3-(2-sulfoethyl)phenyl]amino]carbonyl]glycyl-N2-(3-methoxyphenyl)-N-methyl-N-phenyl-(9CI) | RP 73870 |
|---|
| Type | n/a |
|---|
| Emp. Form. | C26H27N3O7S |
|---|
| Mol. Mass. | 525.573 |
|---|
| SMILES | COc1cccc(c1)N(C(=O)CNC(=O)c1cccc(CCS(O)(=O)=O)c1)C(=O)N(C)c1ccccc1 |
|---|
| Structure | 
|
|---|
Search and Browse
