| Reaction Details |
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 | Report a problem with these data |
| Target | Somatostatin receptor type 2 |
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| Ligand | BDBM82459 |
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| Substrate/Competitor | n/a |
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| Ki | 45.70±n/a nM |
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| Comments | PDSP_387 |
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| Citation |  Hoyer, D; Lübbert, H; Bruns, C Molecular pharmacology of somatostatin receptors. Naunyn Schmiedebergs Arch Pharmacol350:441-53 (1994) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Somatostatin receptor type 2 |
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| Name: | Somatostatin receptor type 2 |
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| Synonyms: | SOMATOSTATIN SST2 | SSR2_MOUSE | Smstr2 | Somatostatin receptor | Somatostatin receptor 2 | Somatostatin receptor type 2 | Sst2 | Sstr2 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 41234.26 |
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| Organism: | MOUSE |
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| Description: | SOMATOSTATIN SST2 SSTR2 MOUSE::P30875 |
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| Residue: | 369 |
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| Sequence: | MEMSSEQLNGSQVWVSSPFDLNGSLGPSNGSNQTEPYYDMTSNAVLTFIYFVVCVVGLCG
NTLVIYVILRYAKMKTITNIYILNLAIADELFMLGLPFLAMQVALVHWPFGKAICRVVMT
VDGINQFTSIFCLTVMSIDRYLAVVHPIKSAKWRRPRTAKMINVAVWCVSLLVILPIMIY
AGLRSNQWGRSSCTINWPGESGAWYTGFIIYAFILGFLVPLTIICLCYLFIIIKVKSSGI
RVGSSKRKKSEKKVTRMVSIVVAVFIFCWLPFYIFNVSSVSVAISPTPALKGMFDFVVIL
TYANSCANPILYAFLSDNFKKSFQNVLCLVKVSGTEDGERSDSKQDKSRLNETTETQRTL
LNGDLQTSI
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| BDBM82459 |
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| n/a |
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| Name | BDBM82459 |
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| Synonyms: | BIM 23058 | BIM-23058 | D-Phe-L-Phe-L-Tyr-D-Trp-L-Lys-L-Val-L-Phe-L-Thr-NH2 |
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| Type | Small organic molecule |
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| Emp. Form. | C62H77N11O10 |
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| Mol. Mass. | 1136.3425 |
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| SMILES | CC(C)[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](N)Cc1ccccc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H]([C@@H](C)O)C(N)=O |
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| Structure | 
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