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TargetSomatostatin receptor type 4
LigandBDBM50065453
Substrate/Competitorn/a
Ki 1000±n/a nM
CommentsPDSP_1035
Citation Hoyer, DLübbert, HBruns, C Molecular pharmacology of somatostatin receptors. Naunyn Schmiedebergs Arch Pharmacol350:441-53 (1994) [PubMed]  Article
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Somatostatin receptor type 4
Name:Somatostatin receptor type 4
Synonyms:SS-4-R | SS4-R | SS4R | SSR4_MOUSE | Smstr4 | Sstr4
Type:PROTEIN
Mol. Mass.:41937.48
Organism:Mus musculus
Description:ChEMBL_833920
Residue:385
Sequence:
MNAPATLPPGVEDTTWTPGINASWAPDEEEEDAMGSDGTGTAGMVTIQCIYALVCLVGLV
GNALVIFVILRYAKMKTATNIYLLNLAVADELFMLSVPFARSAAALRHWPFGAVLCRAVL
SVDGLNMFTSVFCLTVLSVDRYVAVVHPLATATYRRPSVAKLINLGVWLASLLVTLPIAV
FADTRPARGGEAVACNLHWPHPAWSAVFVIYTFLLGFLPPVLAIGLCYLLIVGKMRAVAL
AGGWQQRRRSEKKITRLVLMVVTVFVLCWMPFYVVQLLNLFVTSLDATVNHVSLILSYAN
SCANPILYGFLSDNFRRSFQRVLCLRCCLLETTGGAEEEPLDYYATALKSRGGAGCICPP
LPCQQEPVQAEPGCKQVPFTKTTTF
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BDBM50065453
n/a
NameBDBM50065453
Synonyms:(5S,8S,11S,14R,17S,19aS)-11-(4-Amino-butyl)-5,17-dibenzyl-8-((R)-1-hydroxy-ethyl)-14-(1H-indol-3-ylmethyl)-tetradecahydro-3a,6,9,12,15,18-hexaaza-cyclopentacyclooctadecene-4,7,10,13,16,19-hexaone | CHEMBL421362 | L-361,301 | L-363,301 | L-363301
TypeSmall organic molecule
Emp. Form.C44H54N8O7
Mol. Mass.806.949
SMILESC[C@@H](O)[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H]2CCCN2C(=O)[C@H](Cc2ccccc2)NC1=O
Structure
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