| Reaction Details |
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 | Report a problem with these data |
| Target | Alpha-2B adrenergic receptor |
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| Ligand | BDBM81773 |
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| Substrate/Competitor | n/a |
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| Ki | 0.47±n/a nM |
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| Comments | PDSP_340 |
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| Citation |  O'Rourke, MF; Blaxall, HS; Iversen, LJ; Bylund, DB Characterization of [3H]RX821002 binding to alpha-2 adrenergic receptor subtypes. J Pharmacol Exp Ther268:1362-7 (1994) [PubMed] |
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| More Info.: | Get all data from this article |
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| Alpha-2B adrenergic receptor |
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| Name: | Alpha-2B adrenergic receptor |
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| Synonyms: | ADA2B_DIDVI | ADRA2B | Alpha-2B adrenergic receptor | adrenergic Alpha2 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 41875.91 |
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| Organism: | OPOSSUM |
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| Description: | adrenergic Alpha2 0 OPOSSUM::O77715 |
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| Residue: | 382 |
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| Sequence: | AIAAVITFLILFTIFGNALVILAVLTSRSLRAPQNLFLVSLAAADILVATLIIPFSLANE
LLGYWYFRHTWCEVYLALDVLFCTSSIVHLCAISLDRYWSVSRALEYNSKRTPRRIKGII
LTVWLIAAFISLPPLIYKGDKGKKPGGRPQCKLNEEAWYILSSSIGSFFAPCLIMILVYL
RIYLIAKRRNRQGPHGKQAPGDGDTGPSALGGTSTISKLPPSILPAVGEANGHSKPPGER
EGGEQMGDPTSPSTPPNQSSVGPEDGSQKQEEEEEEEEEEEEECGPPAPPTSSSLQGTPN
FQPSQGSQVLATLRGQVLLARGPASLGLQPWRRRTQMNREKRFTFVLAVVIGVFVLCWFP
FFFSYSLGAICPQHCKVPHGLF
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| BDBM81773 |
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| n/a |
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| Name | BDBM81773 |
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| Synonyms: | BAM 1303 | BAM-1303 | CAS_115219-10-8 |
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| Type | Small organic molecule |
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| Emp. Form. | C25H25BrN4 |
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| Mol. Mass. | 461.397 |
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| SMILES | CN1C[C@H](Cn2ccnc2-c2ccccc2)C[C@H]2[C@H]1Cc1c(Br)[nH]c3cccc2c13 |r| |
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| Structure | 
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