Reaction Details |
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Target | Melatonin receptor type 1A |
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Ligand | BDBM9019 |
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Substrate/Competitor | n/a |
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Ki | 0.24±n/a nM |
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Comments | PDSP_1189 |
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Citation | Reppert, SM; Weaver, DR; Ebisawa, T Cloning and characterization of a mammalian melatonin receptor that mediates reproductive and circadian responses. Neuron13:1177-85 (1994) [PubMed] Article |
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More Info.: | Get all data from this article |
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Melatonin receptor type 1A |
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Name: | Melatonin receptor type 1A |
Synonyms: | MTNR1A | MTR1A_SHEEP | Melatonin | Melatonin receptor type 1A |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 40421.02 |
Organism: | Sheep |
Description: | Melatonin 0 Sheep::P48040 |
Residue: | 366 |
Sequence: | MAGRLWGSPGGTPKGNGSSALLNVSQAAPGAGDGVRPRPSWLAATLASILIFTIVVDIVG
NLLVVLSVYRNKKLRNAGNVFVVSLAVADLLVAVYPYPLALASIVNNGWSLSSLHCQLSG
FLMGLSVIGSVFSITGIAINRYCCICHSLRYGKLYSGTNSLCYVFLIWTLTLVAIVPNLC
VGTLQYDPRIYSCTFTQSVSSAYTIAVVVFHFIVPMLVVVFCYLRIWALVLQVRWKVKPD
NKPKLKPQDFRNFVTMFVVFVLFAICWAPLNFIGLVVASDPASMAPRIPEWLFVASYYMA
YFNSCLNAIIYGLLNQNFRQEYRKIIVSLCTTKMFFVDSSNHVADRIKRKPSPLIANHNL
IKVDSV
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BDBM9019 |
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n/a |
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Name | BDBM9019 |
Synonyms: | CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]acetamide |
Type | Small organic molecule |
Emp. Form. | C13H16N2O2 |
Mol. Mass. | 232.2783 |
SMILES | COc1ccc2[nH]cc(CCNC(C)=O)c2c1 |
Structure |
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