| Reaction Details |
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 | Report a problem with these data |
| Target | Hrh3 protein |
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| Ligand | BDBM82510 |
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| Substrate/Competitor | n/a |
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| Ki | 76±n/a nM |
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| Comments | PDSP_1481 |
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| Citation |  Ligneau, X; Garbarg, M; Vizuete, ML; Diaz, J; Purand, K; Stark, H; Schunack, W; Schwartz, JC [125I]iodoproxyfan, a new antagonist to label and visualize cerebral histamine H3 receptors. J Pharmacol Exp Ther271:452-9 (1994) [PubMed] |
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| More Info.: | Get all data from this article |
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| Hrh3 protein |
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| Name: | Hrh3 protein |
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| Synonyms: | HISTAMINE H3 | HRH3 | Hrh3 protein |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 37860.96 |
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| Organism: | RAT |
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| Description: | Q5PPG3 |
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| Residue: | 344 |
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| Sequence: | MERAPPDGLMNASGTLAGEAAAAGGARGFSAAWTAVLAALMALLIVATVLGNALVMLAFV
ADSSLRTQNNFFLLNLAISDFLVGAFCIPLYVPYVLTGRWTFGRGLCKLWLVVDYLLCAS
SVFNIVLISYDRFLSVTRAVSYRAQQGDTRRAVRKMALVWVLAFLLYGPAILSWEYLSGG
SSIPEGHCYAEFFYNWYFLITASTLEFFTPFLSVTFFNLSIYLNIQRRTRLRLDGGREAG
PEPPPDAQPSPPPAPPSCWGCWPKGHGEAMPLHRGSKPSASSASLEKRMKMVSQSITQRF
RLSRDKKVAKSLAIIVSIFGLCWAPYTLLMIIRAACHGRCIPDY
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| BDBM82510 |
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| n/a |
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| Name | BDBM82510 |
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| Synonyms: | Phenylbutanoylhistamine |
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| Type | Small organic molecule |
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| Emp. Form. | C15H19N3O |
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| Mol. Mass. | 257.3309 |
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| SMILES | CCCC(=O)NCCc1cnc([nH]1)-c1ccccc1 |
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| Structure | 
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