| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Alpha-2A adrenergic receptor |
|---|
| Ligand | BDBM50030623 |
|---|
| Substrate/Competitor | n/a |
|---|
| Ki | 35±n/a nM |
|---|
| Comments | PDSP_1716 |
|---|
| Citation |  O'Rourke, MF; Iversen, LJ; Lomasney, JW; Bylund, DB Species orthologs of the alpha-2A adrenergic receptor: the pharmacological properties of the bovine and rat receptors differ from the human and porcine receptors. J Pharmacol Exp Ther271:735-40 (1994) [PubMed] |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| Alpha-2A adrenergic receptor |
|---|
| Name: | Alpha-2A adrenergic receptor |
|---|
| Synonyms: | Alpha-2A adrenergic receptor | adrenergic Alpha2 | adrenergic Alpha2A |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 48998.96 |
|---|
| Organism: | PIG |
|---|
| Description: | adrenergic Alpha2 0 PIG::P18871 |
|---|
| Residue: | 450 |
|---|
| Sequence: | MGSLQPEAGNASWNGTEAPGGGARATPYSLQVTLTLVCLAGLLMLFTVFGNVLVIIAVFT
SRALKAPQNLFLVSLASADILVATLVIPFSLANEVMGYWYFGKAWCEIYLALDVLFCTSS
IVHLCAISLDRYWSITQAIEYNLKRTPRRIKAIIVTVWVISAVISFPPLISIEKKAGGGG
QQPAEPRCEINDQKWYVISSCIGSFFAPCLIMILVYVRIYQIAKRRTRVPPSRRGPDAAA
ALPGGAERRPNGLGPERGVGRVGAEAEPLPVQLNGAPGEPAPAGPRDADGLDLEESSSSE
HAERPPGPRRSERGPRAKSKARASQVKPGDSLPRRGPGAPGPGAPATGAGEERGGVAKAS
RWRGRQNREKRFTFVLAVVIGVFVVCWFPFFFTYTLTAVGCSVPPTLFKFFFWFGYCNSS
LNPVIYTIFNHDFRRAFKKILCRGDRKRIV
|
|
|
|---|
| BDBM50030623 |
|---|
| n/a |
|---|
| Name | BDBM50030623 |
|---|
| Synonyms: | 6-Chloro-3-methyl-9-(3-methyl-but-2-enyloxy)-2,3,4,5-tetrahydro-1H-benzo[d]azepine | CHEMBL114166 | SK&F-104078 | SK-104078 | SKF 104078 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C16H22ClNO |
|---|
| Mol. Mass. | 279.805 |
|---|
| SMILES | [#6]-[#7]-1-[#6]-[#6]-c2c(Cl)ccc(-[#8]-[#6]\[#6]=[#6](\[#6])-[#6])c2-[#6]-[#6]-1 |
|---|
| Structure | 
|
|---|
Search and Browse
