| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Alpha-2A adrenergic receptor |
|---|
| Ligand | BDBM81444 |
|---|
| Substrate/Competitor | n/a |
|---|
| Ki | 13.2±n/a nM |
|---|
| Comments | PDSP_1955 |
|---|
| Citation |  O'Rourke, MF; Iversen, LJ; Lomasney, JW; Bylund, DB Species orthologs of the alpha-2A adrenergic receptor: the pharmacological properties of the bovine and rat receptors differ from the human and porcine receptors. J Pharmacol Exp Ther271:735-40 (1994) [PubMed] |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| Alpha-2A adrenergic receptor |
|---|
| Name: | Alpha-2A adrenergic receptor |
|---|
| Synonyms: | ADA2A_BOVIN | ADRA2A | Alpha-2A adrenergic receptor | Alpha-2A adrenoceptor | Alpha-2A adrenoreceptor | Alpha-2AAR | Alpha-2D adrenergic receptor | Alpha-2Da adrenergic receptor | Cerebral cortex alpha adrenergic receptor | adrenergic Alpha2A | adrenergic Alpha2D |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 49275.13 |
|---|
| Organism: | BOVINE |
|---|
| Description: | adrenergic Alpha2 0 BOVINE::Q28838 |
|---|
| Residue: | 452 |
|---|
| Sequence: | MGSLQPDAGNASWNGTEAPGGGARATPYSLQVTLTLVCLAGLLMLFTVFGNVLVIIAVFT
SRALKAPQNLFLVSLASADILVATLVIPFSLANEVMGYWYFGKAWCEIYLALDVLFCTSS
IVHLCAISLDRYWSITQAIEYNLKRTPRRIKAIIVTVWVISAVISFPPLISFEKKRGRSG
QPSAEPRCEINDQKWYVISSSIGSFFAPCLIMILVYVRIYQIAKRRTRVPPSRRGPDATA
AELPGSAERRPNGLGPERGGVGPVGAEVESLQVQLNGAPGEPAPAGAGADALDLEESSSS
EHAERPPGSRRSERGPRAKGKARASQVKPGDSLPRRGPGATGLGAPTAGPAEERSGGGAK
ASRWRGRQNREKRFTFVLAVVIGVFVVCWFPFFFTYTLTAIGCPVPPTLFKFFFWFGYCN
SSLNPVIYTIFNHDFRRAFKKILCRGDRKRIV
|
|
|
|---|
| BDBM81444 |
|---|
| n/a |
|---|
| Name | BDBM81444 |
|---|
| Synonyms: | CAS_185453 | NSC_185453 | WB 4101 | WB-4101 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C25H27NO5 |
|---|
| Mol. Mass. | 421.4856 |
|---|
| SMILES | COc1cccc(OC)c1OCCNCC1Oc2ccccc2OC1c1ccccc1 |
|---|
| Structure | 
|
|---|
Search and Browse
