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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | 5-hydroxytryptamine receptor 7 | ||
| Ligand | BDBM50031942 | ||
| Substrate/Competitor | n/a | ||
| Ki | 13.48±n/a nM | ||
| Comments | PDSP_1230 | ||
| Citation |  Boess, FG; Martin, IL Molecular biology of 5-HT receptors. Neuropharmacology33:275-317 (1994) [PubMed] Article | ||
| More Info.: | Get all data from this article | ||
| 5-hydroxytryptamine receptor 7 | |||
| Name: | 5-hydroxytryptamine receptor 7 | ||
| Synonyms: | 5-HT-7 | 5-HT-X | 5-HT7 | 5-HT7L | 5-HT7S | 5-Hydroxytryptamine receptor 7 (5-HT7) | 5-hydroxytryptamine receptor 7 | 5-hydroxytryptamine receptor 7 (5-HT-7) | 5HT7R_RAT | Adrenergic Alpha | GPRFO | Htr7 | Serotonin (5-HT) receptor | Serotonin Receptor 7 | ||
| Type: | G Protein-Coupled Receptor (GPCR) | ||
| Mol. Mass.: | 49852.62 | ||
| Organism: | Rattus norvegicus (rat) | ||
| Description: | Rat cloned 5-HT7R. | ||
| Residue: | 448 | ||
| Sequence: |
| ||
| BDBM50031942 | |||
| n/a | |||
| Name | BDBM50031942 | ||
| Synonyms: | (6aR,9R)-4,6a,7-Trimethyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid (1-hydroxymethyl-propyl)-amide | (6aR,9R)-4,7-Dimethyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid ((S)-1-hydroxymethyl-propyl)-amide | (6aR,9R)-4-Methyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid (1-hydroxymethyl-propyl)-amide | (6aR,9R)-5,7-Dimethyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid diethylamide | (methylsergide)4,7-Dimethyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid (1-hydroxymethyl-propyl)-amide | 4,7-Dimethyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid (1-hydroxymethyl-propyl)-amide | CHEMBL1065 | METHYSERGIDE | Sansert | ||
| Type | Small organic molecule | ||
| Emp. Form. | C21H27N3O2 | ||
| Mol. Mass. | 353.458 | ||
| SMILES | CC[C@@H](CO)NC(=O)[C@H]1CN(C)[C@@H]2Cc3cn(C)c4cccc(C2=C1)c34 |r,c:24| | ||
| Structure | 
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