| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1 |
|---|
| Ligand | BDBM52287 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Dose Response confirmation of uHTS hits for Scp-1 phosphatase using a colorimetric assay |
|---|
| IC50 | 1595±171 nM |
|---|
| Citation |  PubChem, PC Dose Response confirmation of uHTS hits for Scp-1 phosphatase using a colorimetric assay PubChem Bioassay(2011)[AID] |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1 |
|---|
| Name: | Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1 |
|---|
| Synonyms: | CTDS1_HUMAN | CTDSP1 | NIF3 | NLIIF | SCP1 | carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1 isoform 1 |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 29199.89 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | gi_10864009 |
|---|
| Residue: | 261 |
|---|
| Sequence: | MDSSAVITQISKEEARGPLRGKGDQKSAASQKPRSRGILHSLFCCVCRDDGEALPAHSGA
PLLVEENGAIPKQTPVQYLLPEAKAQDSDKICVVIDLDETLVHSSFKPVNNADFIIPVEI
DGVVHQVYVLKRPHVDEFLQRMGELFECVLFTASLAKYADPVADLLDKWGAFRARLFRES
CVFHRGNYVKDLSRLGRDLRRVLILDNSPASYVFHPDNAVPVASWFDNMSDTELHDLLPF
FEQLSRVDDVYSVLRQPRPGS
|
|
|
|---|
| BDBM52287 |
|---|
| n/a |
|---|
| Name | BDBM52287 |
|---|
| Synonyms: | 4-[3-(5-Furan-2-yl-2H-pyrazol-3-yl)-5-mercapto-[1,2,4]triazol-4-yl]-benzoic acid | 4-[3-[5-(2-furanyl)-1H-pyrazol-3-yl]-5-sulfanylidene-1H-1,2,4-triazol-4-yl]benzoic acid | 4-[3-[5-(2-furyl)-1H-pyrazol-3-yl]-5-thioxo-1H-1,2,4-triazol-4-yl]benzoic acid | 4-[3-[5-(furan-2-yl)-1H-pyrazol-3-yl]-5-sulfanylidene-1H-1,2,4-triazol-4-yl]benzoic acid | MLS000551487 | SMR000145412 | cid_1839198 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C16H11N5O3S |
|---|
| Mol. Mass. | 353.355 |
|---|
| SMILES | OC(=O)c1ccc(cc1)-n1c(n[nH]c1=S)-c1cc([nH]n1)-c1ccco1 |
|---|
| Structure | 
|
|---|
Search and Browse
