Ki Summary

Reaction Details

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Target

Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1

Ligand

BDBM82835

Substrate/Competitor

n/a

Meas. Tech.

Dose Response confirmation of uHTS hits for Scp-1 phosphatase using a colorimetric assay

IC50

1830±88 nM

Citation

PubChem, PC Dose Response confirmation of uHTS hits for Scp-1 phosphatase using a colorimetric assay PubChem Bioassay(2011)[AID]

More Info.:

Get all data from this article, Assay Method

Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1

Name:

Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1

Synonyms:

Type:

Enzyme Catalytic Domain

Mol. Mass.:

29199.89

Organism:

Homo sapiens (Human)

Description:

gi_10864009

Residue:

261

Sequence:

MDSSAVITQISKEEARGPLRGKGDQKSAASQKPRSRGILHSLFCCVCRDDGEALPAHSGA
PLLVEENGAIPKQTPVQYLLPEAKAQDSDKICVVIDLDETLVHSSFKPVNNADFIIPVEI
DGVVHQVYVLKRPHVDEFLQRMGELFECVLFTASLAKYADPVADLLDKWGAFRARLFRES
CVFHRGNYVKDLSRLGRDLRRVLILDNSPASYVFHPDNAVPVASWFDNMSDTELHDLLPF
FEQLSRVDDVYSVLRQPRPGS

BDBM82835

n/a

Name

BDBM82835

Synonyms:

4-(5,5-dimethyl-3-morpholin-4-yl-cyclohex-2-en-1-ylidene)-2,6-dimethyl-morpholin-4-ium;iodide | 4-(5,5-dimethyl-3-morpholin-4-ylcyclohex-2-en-1-ylidene)-2,6-dimethylmorpholin-4-ium;iodide | 4-(5,5-dimethyl-3-morpholino-cyclohex-2-en-1-ylidene)-2,6-dimethyl-morpholin-4-ium;iodide | 4-[5,5-dimethyl-3-(4-morpholinyl)-1-cyclohex-2-enylidene]-2,6-dimethylmorpholin-4-ium;iodide | MLS001032833 | SMR000363499 | cid_16196366

Type

Small organic molecule

Emp. Form.

C18H31N2O2

Mol. Mass.

307.4504

SMILES

[#6]-[#6]-1-[#6]\[#7+](-[#6]-[#6](-[#6])-[#8]-1)=[#6]-1/[#6]C([#6])([#6])[#6]-[#6](=[#6]-1)-[#7]-1-[#6]-[#6]-[#8]-[#6]-[#6]-1 |c:15|

Structure