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TargetCarboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1
LigandBDBM59546
Substrate/Competitorn/a
Meas. Tech.Dose Response confirmation of uHTS hits for Scp-1 phosphatase using a colorimetric assay
IC50 1988±246 nM
Citation PubChem, PC Dose Response confirmation of uHTS hits for Scp-1 phosphatase using a colorimetric assay PubChem Bioassay(2011)[AID]
More Info.:Get all data from this article,  Assay Method
 
Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1
Name:Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1
Synonyms:CTDS1_HUMAN | CTDSP1 | NIF3 | NLIIF | SCP1 | carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1 isoform 1
Type:Enzyme Catalytic Domain
Mol. Mass.:29199.89
Organism:Homo sapiens (Human)
Description:gi_10864009
Residue:261
Sequence:
MDSSAVITQISKEEARGPLRGKGDQKSAASQKPRSRGILHSLFCCVCRDDGEALPAHSGA
PLLVEENGAIPKQTPVQYLLPEAKAQDSDKICVVIDLDETLVHSSFKPVNNADFIIPVEI
DGVVHQVYVLKRPHVDEFLQRMGELFECVLFTASLAKYADPVADLLDKWGAFRARLFRES
CVFHRGNYVKDLSRLGRDLRRVLILDNSPASYVFHPDNAVPVASWFDNMSDTELHDLLPF
FEQLSRVDDVYSVLRQPRPGS
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  Blast E-value cutoff:
BDBM59546
n/a
NameBDBM59546
Synonyms:3-[7-(2-chlorobenzyl)oxy-2-keto-4,8-dimethyl-chromen-3-yl]propionic acid | 3-[7-[(2-chlorophenyl)methoxy]-4,8-dimethyl-2-oxidanylidene-chromen-3-yl]propanoic acid | 3-[7-[(2-chlorophenyl)methoxy]-4,8-dimethyl-2-oxo-1-benzopyran-3-yl]propanoic acid | 3-[7-[(2-chlorophenyl)methoxy]-4,8-dimethyl-2-oxochromen-3-yl]propanoic acid | MLS001213288 | SMR000540578 | cid_1801772
TypeSmall organic molecule
Emp. Form.C21H19ClO5
Mol. Mass.386.826
SMILESCc1c(OCc2ccccc2Cl)ccc2c(C)c(CCC(O)=O)c(=O)oc12
Structure
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