Reaction Details |
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Target | Phospholipase A2 |
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Ligand | BDBM33185 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Dose response counterscreen of uHTS hits for ATG4B inhibitors in a Phospholipase A2 assay |
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IC50 | 34700±n/a nM |
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Citation | PubChem, PC Dose response counterscreen of uHTS hits for ATG4B inhibitors in a Phospholipase A2 assay PubChem Bioassay(2011)[AID] |
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More Info.: | Get all data from this article, Assay Method |
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Phospholipase A2 |
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Name: | Phospholipase A2 |
Synonyms: | Group IB phospholipase A2 | PA21B_HUMAN | PLA2 | PLA2A | PLA2G1B | PPLA2 | Phosphatidylcholine 2-acylhydrolase 1B | Phospholipase A2 (PLA2) | Phospholipase A2 group 1B | phospholipase A2 precursor |
Type: | Protein |
Mol. Mass.: | 16364.13 |
Organism: | Homo sapiens (Human) |
Description: | P04054 |
Residue: | 148 |
Sequence: | MKLLVLAVLLTVAAADSGISPRAVWQFRKMIKCVIPGSDPFLEYNNYGCYCGLGGSGTPV
DELDKCCQTHDNCYDQAKKLDSCKFLLDNPYTHTYSYSCSGSAITCSSKNKECEAFICNC
DRNAAICFSKAPYNKAHKNLDTKKYCQS
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BDBM33185 |
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n/a |
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Name | BDBM33185 |
Synonyms: | 4-({(4Z)-1-oxo-4-[(phenylsulfonyl)imino]-1,4-dihydronaphthalen-2-yl}amino)benzoic acid | 4-[(4-besylimino-1-keto-2-naphthyl)amino]benzoic acid | 4-[[(4Z)-4-besylimino-1-keto-2-naphthyl]amino]benzoic acid | 4-[[1-oxidanylidene-4-(phenylsulfonylimino)naphthalen-2-yl]amino]benzoic acid | 4-[[4-(benzenesulfonylimino)-1-oxo-2-naphthalenyl]amino]benzoic acid | 4-[[4-(benzenesulfonylimino)-1-oxonaphthalen-2-yl]amino]benzoic acid | MLS000686314 | SMR000313157 | cid_4053104 |
Type | Small organic molecule |
Emp. Form. | C23H16N2O5S |
Mol. Mass. | 432.449 |
SMILES | OC(=O)c1ccc(NC2=CC(=NS(=O)(=O)c3ccccc3)c3ccccc3C2=O)cc1 |w:11.11,t:8| |
Structure |
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