| Reaction Details |
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 | Report a problem with these data |
| Target | Somatostatin receptor type 3 |
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| Ligand | BDBM84619 |
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| Substrate/Competitor | n/a |
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| Ki | 11±n/a nM |
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| Comments | PDSP_392 |
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| Citation |  Raynor, K; Murphy, WA; Coy, DH; Taylor, JE; Moreau, JP; Yasuda, K; Bell, GI; Reisine, T Cloned somatostatin receptors: identification of subtype-selective peptides and demonstration of high affinity binding of linear peptides. Mol Pharmacol43:838-44 (1993) [PubMed] |
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| More Info.: | Get all data from this article |
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| Somatostatin receptor type 3 |
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| Name: | Somatostatin receptor type 3 |
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| Synonyms: | SOMATOSTATIN SST3 | SS3R | SSR-28 | SSR3_MOUSE | Smstr3 | Somatostatin receptor | Somatostatin receptor 3 | Somatostatin receptor type 3 | Sstr3 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 47225.49 |
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| Organism: | MOUSE |
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| Description: | SOMATOSTATIN SST3 SSTR3 MOUSE::P30935 |
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| Residue: | 428 |
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| Sequence: | MATVTYPSSEPTTLDPGNASSTWPLDTTLGNTSAGASLTGLAVSGILISLVYLVVCVVGL
LGNSLVIYVVLRHTSSPSVTSVYILNLALADELFMLGLPFLAAQNALSYWPFGSLMCRLV
MAVDGINQFTSIFCLTVMSVDRYLAVVHPTRSARWRTAPVARTVSAAVWVASAVVVLPVV
VFSGVPRGMSTCHMQWPEPAAAWRTAFIIYTAALGFFGPLLVICLCYLLIVVKVRSTTRR
VRAPSCQWVQAPACQRRRRSERRVTRMVVAVVALFVLCWMPFYLLNIVNVVCPLPEEPAF
FGLYFLVVALPYANSCANPILYGFLSYRFKQGFRRILLRPSRRIRSQEPGSGPPEKTEEE
EDEEEEERREEEERRMQRGQEMNGRLSQIAQAGTSGQQPRPCTGTAKEQQLLPQEATAGD
KASTLSHL
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| BDBM84619 |
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| n/a |
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| Name | BDBM84619 |
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| Synonyms: | BIM 23065 | CAS_150155-63-8 | L-Threoninamide,3-(2-naphthalenyl)-D-alanyl-4-chloro-L-phenylalanyl-L-tyrosyl-D-tryptophyl-L-lysyl-L-threonyl-L-phenylalanyl-(9CI) |
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| Type | Small organic molecule |
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| Emp. Form. | C69H83ClN12O13 |
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| Mol. Mass. | 1323.923 |
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| SMILES | C[C@@H](O)[C@H](NC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](CCCCN)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(Cc1ccc(O)cc1)NC(=O)[C@H](Cc1ccc(Cl)cc1)NC(=O)[C@H](N)Cc1ccc2ccccc2c1)C(C)O)C(C)O)C(N)=O |r| |
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| Structure | 
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