| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Mu-type opioid receptor |
|---|
| Ligand | BDBM50000571 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_146696 (CHEMBL753773) |
|---|
| Ki | 140±n/a nM |
|---|
| Citation |  Froimowitz, M; Pick, CG; Pasternak, GW Phenylmorphans and analogues: opioid receptor subtype selectivity and effect of conformation on activity. J Med Chem35:1521-5 (1992) [PubMed] |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Mu-type opioid receptor |
|---|
| Name: | Mu-type opioid receptor |
|---|
| Synonyms: | MOR-1 | Mu opioid receptor | OPIATE Mu | OPRM1 | OPRM_BOVIN |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 45038.37 |
|---|
| Organism: | CALF |
|---|
| Description: | OPIATE Mu 2 0 CALF::P79350 |
|---|
| Residue: | 401 |
|---|
| Sequence: | MDSGAVPTNASNCTDPFTHPSSCSPAPSPSSWVNFSHLEGNLSDPCGPNRTELGGSDRLC
PSAGSPSMITAIIIMALYSIVCVVGLFGNFLVMYVIVRYTKMKTATNIYIFNLALADALA
TSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALD
LRTPRNAKIINICNWILSSAIGLPVMFMATTKYRQGSIDCTLTFSHPTWYWENLLKICVF
IFAFIMPILIITVCYGLMILRLKSVRMLSGSKEKDRNLRRITRMVLVVVAVFIVCWTPIH
IYVIIKALITIPETTFQTVSWHFCIALGYTNSCLNPVLYAFLDENFKRCFREFCIPTSST
IEQQNSTRIRQNTRDHPSTANTVDRTNHQLENLEAETTPLP
|
|
|
|---|
| BDBM50000571 |
|---|
| n/a |
|---|
| Name | BDBM50000571 |
|---|
| Synonyms: | 3-(2,9-Dimethyl-2-aza-bicyclo[3.3.1]non-5-yl)-phenol | 5-(3-Hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]nonan-9-ol | CHEMBL287726 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C16H23NO |
|---|
| Mol. Mass. | 245.3599 |
|---|
| SMILES | C[C@@H]1C2CCCC1(CCN2C)c1cccc(O)c1 |TLB:10:9:1:5.3.4,THB:0:1:9.7.8:5.3.4| |
|---|
| Structure | 
|
|---|
Search and Browse
