Reaction Details |
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Target | Neuropeptide Y receptor type 4 |
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Ligand | BDBM50240829 |
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Substrate/Competitor | n/a |
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Meas. Tech. | ChEMBL_1669006 (CHEMBL4018894) |
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Ki | 0.063096±n/a nM |
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Citation | Schubert, M; Stichel, J; Du, Y; Tough, IR; Sliwoski, G; Meiler, J; Cox, HM; Weaver, CD; Beck-Sickinger, AG Identification and Characterization of the First Selective Y J Med Chem60:7605-7612 (2017) [PubMed] Article |
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More Info.: | Get all data from this article, Assay Method |
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Neuropeptide Y receptor type 4 |
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Name: | Neuropeptide Y receptor type 4 |
Synonyms: | NPY-Y4 | NPY4-R | NPY4R | NPY4R_HUMAN | PP1 | PPYR1 | Pancreatic polypeptide receptor 1 |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 42207.58 |
Organism: | Homo sapiens (Human) |
Description: | NPY-Y4 PPYR1 HUMAN::P50391 |
Residue: | 375 |
Sequence: | MNTSHLLALLLPKSPQGENRSKPLGTPYNFSEHCQDSVDVMVFIVTSYSIETVVGVLGNL
CLMCVTVRQKEKANVTNLLIANLAFSDFLMCLLCQPLTAVYTIMDYWIFGETLCKMSAFI
QCMSVTVSILSLVLVALERHQLIINPTGWKPSISQAYLGIVLIWVIACVLSLPFLANSIL
ENVFHKNHSKALEFLADKVVCTESWPLAHHRTIYTTFLLLFQYCLPLGFILVCYARIYRR
LQRQGRVFHKGTYSLRAGHMKQVNVVLVVMVVAFAVLWLPLHVFNSLEDWHHEAIPICHG
NLIFLVCHLLAMASTCVNPFIYGFLNTNFKKEIKALVLTCQQSAPLEESEHLPLSTVHTE
VSKGSLRLSGRSNPI
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BDBM50240829 |
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n/a |
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Name | BDBM50240829 |
Synonyms: | CHEMBL3559801 |
Type | Small organic molecule |
Emp. Form. | C16H24O2 |
Mol. Mass. | 248.3606 |
SMILES | CC(C)(C)c1ccc(OC2CCCCC2O)cc1 |
Structure |
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