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TargetNeuropeptide Y receptor type 4
LigandBDBM50240829
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1669006 (CHEMBL4018894)
Ki 0.063096±n/a nM
Citation Schubert, MStichel, JDu, YTough, IRSliwoski, GMeiler, JCox, HMWeaver, CDBeck-Sickinger, AG Identification and Characterization of the First Selective Y J Med Chem60:7605-7612 (2017) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Neuropeptide Y receptor type 4
Name:Neuropeptide Y receptor type 4
Synonyms:NPY-Y4 | NPY4-R | NPY4R | NPY4R_HUMAN | PP1 | PPYR1 | Pancreatic polypeptide receptor 1
Type:Enzyme Catalytic Domain
Mol. Mass.:42207.58
Organism:Homo sapiens (Human)
Description:NPY-Y4 PPYR1 HUMAN::P50391
Residue:375
Sequence:
MNTSHLLALLLPKSPQGENRSKPLGTPYNFSEHCQDSVDVMVFIVTSYSIETVVGVLGNL
CLMCVTVRQKEKANVTNLLIANLAFSDFLMCLLCQPLTAVYTIMDYWIFGETLCKMSAFI
QCMSVTVSILSLVLVALERHQLIINPTGWKPSISQAYLGIVLIWVIACVLSLPFLANSIL
ENVFHKNHSKALEFLADKVVCTESWPLAHHRTIYTTFLLLFQYCLPLGFILVCYARIYRR
LQRQGRVFHKGTYSLRAGHMKQVNVVLVVMVVAFAVLWLPLHVFNSLEDWHHEAIPICHG
NLIFLVCHLLAMASTCVNPFIYGFLNTNFKKEIKALVLTCQQSAPLEESEHLPLSTVHTE
VSKGSLRLSGRSNPI
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BDBM50240829
n/a
NameBDBM50240829
Synonyms:CHEMBL3559801
TypeSmall organic molecule
Emp. Form.C16H24O2
Mol. Mass.248.3606
SMILESCC(C)(C)c1ccc(OC2CCCCC2O)cc1
Structure
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