Reaction Details |
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Target | Growth hormone-releasing hormone receptor |
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Ligand | BDBM50004976 |
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Substrate/Competitor | n/a |
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Meas. Tech. | ChEBML_72520 |
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IC50 | 1.9±n/a nM |
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Citation | Gaudreau, P; Boulanger, L; Abribat, T Affinity of human growth hormone-releasing factor (1-29)NH2 analogues for GRF binding sites in rat adenopituitary. J Med Chem35:1864-9 (1992) [PubMed] |
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More Info.: | Get all data from this article, Assay Method |
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Growth hormone-releasing hormone receptor |
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Name: | Growth hormone-releasing hormone receptor |
Synonyms: | GHRH receptor | GHRHR_RAT | GRF receptor | Ghrhr | Grfr |
Type: | PROTEIN |
Mol. Mass.: | 51523.38 |
Organism: | Rattus norvegicus |
Description: | ChEMBL_193173 |
Residue: | 464 |
Sequence: | MDSLLWATWVLCLLNLWGVALGHLHLECDFITQLRDDELACLQAAEGTNNSSMGCPGTWD
GLLCWPPTGSGQWVSLPCPEFFSHFGSDPGAVKRDCTITGWSDPFPPYPVACPVPLELLT
EEKSYFSTVKIIYTTGHSISIVALCVAIAILVALRRLHCPRNYIHTQLFATFILKASAVF
LKDAAVFQGDSTDHCSMSTILCKVSVAVSHFATMTNFSWLLAEAVYLSCLLASTSPRSKP
AFWWLVLAGWGLPVLCTGTWVGCKLAFEDTACWDLDDSSPYWWIIKGPIVLSVGVNFGLF
LNIICILLRKLGPAQGGLHTRAQYCNYLLPWSCPLPQVPRERTDLGPSSHEITVQESGTR
NCQLPWRLSKSTLLLIPLFGIHYIIFNFLPDSAGLGIRLPLELGLGSFQGFVVAVLYCFL
NQEVRTEISRKWYGHDPELLPARRTCTEWTTPPRSRVKVLTSEC
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BDBM50004976 |
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n/a |
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Name | BDBM50004976 |
Synonyms: | CHEMBL385308 | GRF-analogues |
Type | Small organic molecule |
Emp. Form. | C157H253N49O41S |
Mol. Mass. | 3515.057 |
SMILES | n/a |
Structure |
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