| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50008888 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_146259 (CHEMBL757483) |
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| Ki | 464±n/a nM |
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| Citation |  Vecchietti, V; Giordani, A; Giardina, G; Colle, R; Clarke, GD (2S)-1-(arylacetyl)-2-(aminomethyl)piperidine derivatives: novel, highly selective kappa opioid analgesics. J Med Chem34:397-403 (1991) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 11165.58 |
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| Organism: | GUINEA PIG |
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| Description: | P97266 |
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| Residue: | 98 |
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| Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
|
|
|
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| BDBM50008888 |
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| n/a |
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| Name | BDBM50008888 |
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| Synonyms: | (threo)2-(3,4-Dichloro-phenyl)-1-[2-(1-methyl-pyrrolidin-2-yl)-piperidin-1-yl]-ethanone(HCl) | 2-(3,4-Dichloro-phenyl)-1-[2-(1-methyl-pyrrolidin-2-yl)-piperidin-1-yl]-ethanone(HCl) | CHEMBL130272 |
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| Type | Small organic molecule |
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| Emp. Form. | C18H24Cl2N2O |
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| Mol. Mass. | 355.302 |
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| SMILES | CN1CCCC1C1CCCCN1C(=O)Cc1ccc(Cl)c(Cl)c1 |
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| Structure | 
|
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