| Reaction Details |
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 | Report a problem with these data |
| Target | Thromboxane A2 receptor |
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| Ligand | BDBM50010077 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_209599 |
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| Kd | 21±n/a nM |
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| Citation |  Misra, RN; Brown, BR; Han, WC; Harris, DN; Hedberg, A; Webb, ML; Hall, SE Interphenylene 7-oxabicyclo[2.2.1]heptane thromboxane A2 antagonists. Semicarbazone omega-chains. J Med Chem34:2882-91 (1991) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Thromboxane A2 receptor |
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| Name: | Thromboxane A2 receptor |
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| Synonyms: | Prostanoid TP receptor | TA2R_HUMAN | TBXA2R | TXA2-R | Thromboxane | Thromboxane A2 receptor | Thromboxane Beta |
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| Type: | Enyzme |
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| Mol. Mass.: | 37445.28 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P21731 |
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| Residue: | 343 |
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| Sequence: | MWPNGSSLGPCFRPTNITLEERRLIASPWFAASFCVVGLASNLLALSVLAGARQGGSHTR
SSFLTFLCGLVLTDFLGLLVTGTIVVSQHAALFEWHAVDPGCRLCRFMGVVMIFFGLSPL
LLGAAMASERYLGITRPFSRPAVASQRRAWATVGLVWAAALALGLLPLLGVGRYTVQYPG
SWCFLTLGAESGDVAFGLLFSMLGGLSVGLSFLLNTVSVATLCHVYHGQEAAQQRPRDSE
VEMMAQLLGIMVVASVCWLPLLVFIAQTVLRNPPAMSPAGQLSRTTEKELLIYLRVATWN
QILDPWVYILFRRAVLRRLQPRLSTRPRSLSLQPQLTQRSGLQ
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| BDBM50010077 |
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| n/a |
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| Name | BDBM50010077 |
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| Synonyms: | 4-[2-(5-oxabicyclo[2.2.1],3-formaldehyde (anilinocarbonyl)hydrazonehept-2-ylmethyl)phenyl]butanoic acid | CHEMBL95867 |
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| Type | Small organic molecule |
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| Emp. Form. | C25H29N3O4 |
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| Mol. Mass. | 435.5155 |
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| SMILES | OC(=O)CCCc1ccccc1CC1C2CCC(O2)C1C=NNC(=O)Nc1ccccc1 |w:21.24,THB:20:19:18:16.15| |
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| Structure | 
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