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TargetAdenosine receptor A2a and A3
LigandBDBM50078423
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1701162
Ki 212±n/a nM
Citation Petrelli RScortichini MKachler SBoccella SCerchia CTorquati IDel Bello FSalvemini DNovellino ELuongo LMaione SJacobson KALavecchia AKlotz KNCappellacci L Exploring the Role of N J Med Chem 60:4327-4341 (2017) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Adenosine receptor A2a and A3
Name:Adenosine receptor A2a and A3
Synonyms:Adenosine A3 receptor
Type:PROTEIN
Mol. Mass.:36643.73
Organism:Rattus norvegicus
Description:ChEMBL_479910
Residue:320
Sequence:
MKANNTTTSALWLQITYITMEAAIGLCAVVGNMLVIWVVKLNRTLRTTTFYFIVSLALAD
IAVGVLVIPLAIAVSLEVQMHFYACLFMSCVLLVFTHASIMSLLAIAVDRYLRVKLTVRY
RTVTTQRRIWLFLGLCWLVSFLVGLTPMFGWNRKVTLELSQNSSTLSCHFRSVVGLDYMV
FFSFITWILIPLVVMCIIYLDIFYIIRNKLSQNLTGFRETRAFYGREFKTAKSLFLVLFL
FALCWLPLSIINFVSYFNVKIPEIAMCLGILLSHANSMMNPIVYACKIKKFKETYFVILR
ACRLCQTSDSLDSNLEQTTE
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50078423
n/a
NameBDBM50078423
Synonyms:CHEMBL3414937
TypeSmall organic molecule
Emp. Form.C12H14ClN9O3
Mol. Mass.367.751
SMILESCCn1nnc(n1)[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)nc(Cl)nc12 |r|
Structure
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