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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Leukotriene B4 receptor 1 | ||
| Ligand | BDBM50013889 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | ChEBML_99660 | ||
| IC50 | 1.9±n/a nM | ||
| Citation |  Gapinski, DM; Mallett, BE; Froelich, LL; Jackson, WT Benzophenone dicarboxylic acid antagonists of leukotriene B4. 2. Structure-activity relationships of the lipophilic side chain. J Med Chem33:2807-13 (1990) [PubMed] | ||
| More Info.: | Get all data from this article, Assay Method | ||
| Leukotriene B4 receptor 1 | |||
| Name: | Leukotriene B4 receptor 1 | ||
| Synonyms: | BLT | BLT1 | BLTR | CMKRL1 | Chemoattractant receptor-like 1 | G-protein coupled receptor 16 | GPR16 | LT4R1_HUMAN | LTB4-R 1 | LTB4R | Leukotriene B4 R1 | Leukotriene B4 receptor | Leukotriene B4 receptor 1 | P2RY7 | P2Y purinoceptor 7 | P2Y7 | ||
| Type: | Enzyme Catalytic Domain | ||
| Mol. Mass.: | 37582.68 | ||
| Organism: | Homo sapiens (Human) | ||
| Description: | Q15722 | ||
| Residue: | 352 | ||
| Sequence: |
| ||
| BDBM50013889 | |||
| n/a | |||
| Name | BDBM50013889 | ||
| Synonyms: | (5S,6Z,8E,10E,12R,14Z)-5,12-dihydroxyicosa-6,8,10,14-tetraenoic acid | (S-(R*,S*-(E,Z,E,Z)))-5,12-Dihydroxy-6,8,10,14-eicosatetraenoic acid | 5,12-Dihete | 5,12-Hete | 5S,12R-dihydroxy-6Z,8E,10E,14Z-eicosatetraenoic acid | CHEMBL65061 | DIHETE 12(s), 5(s) | LTB4 | leukotriene B4 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C20H32O4 | ||
| Mol. Mass. | 336.4657 | ||
| SMILES | CCCCC\C=C/C[C@@H](O)\C=C\C=C\C=C/[C@@H](O)CCCC(O)=O |r| | ||
| Structure | 
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