| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Beta-2 adrenergic receptor |
|---|
| Ligand | BDBM50019968 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEBML_38483 |
|---|
| IC50 | >10000±n/a nM |
|---|
| Citation |  DeWald, HA; Beeson, NW; Hershenson, FM; Wise, LD; Downs, DA; Heffner, TG; Coughenour, LL; Pugsley, TA Synthesis and potential antipsychotic activity of 1H-imidazo[1,2-c]pyrazolo[3,4-e]pyrimidines. J Med Chem31:454-61 (1988) [PubMed] |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Beta-2 adrenergic receptor |
|---|
| Name: | Beta-2 adrenergic receptor |
|---|
| Synonyms: | ADRB2_RAT | Adrb2 | Adrb2r | Adrenergic receptor beta |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 46896.26 |
|---|
| Organism: | Rattus norvegicus |
|---|
| Description: | ChEMBL_38603 |
|---|
| Residue: | 418 |
|---|
| Sequence: | MEPHGNDSDFLLAPNGSRAPGHDITQERDEAWVVGMAILMSVIVLAIVFGNVLVITAIAK
FERLQTVTNYFITSLACADLVMGLAVVPFGASHILMKMWNFGNFWCEFWTSIDVLCVTAS
IETLCVIAVDRYVAITSPFKYQSLLTKNKARVVILMVWIVSGLTSFLPIQMHWYRATHKQ
AIDCYAKETCCDFFTNQAYAIASSIVSFYVPLVVMVFVYSRVFQVAKRQLQKIDKSEGRF
HAQNLSQVEQDGRSGHGLRSSSKFCLKEHKALKTLGIIMGTFTLCWLPFFIVNIVHVIRA
NLIPKEVYILLNWLGYVNSAFNPLIYCRSPDFRIAFQELLCLRRSSSKTYGNGYSSNSNG
RTDYTGEQSAYQLGQEKENELLCEEAPGMEGFVNCQGTVPSLSIDSQGRNCNTNDSPL
|
|
|
|---|
| BDBM50019968 |
|---|
| n/a |
|---|
| Name | BDBM50019968 |
|---|
| Synonyms: | 7-Ethyl-1,3,5-trimethyl-6,7-dihydro-1H-1,2,4,5a,8-pentaaza-as-indacene | CHEMBL143865 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C12H17N5 |
|---|
| Mol. Mass. | 231.2969 |
|---|
| SMILES | CCC1CN2C(=N1)c1c(N=C2C)c(C)nn1C |c:5,10| |
|---|
| Structure | 
|
|---|
Search and Browse
