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TargetGamma-aminobutyric acid receptor subunit gamma-1
LigandBDBM24183
Substrate/Competitorn/a
Meas. Tech.ChEBML_68602
IC50 33±n/a nM
Citation Krogsgaard-Larsen, PNielsen, LFalch, ECurtis, DR GABA agonists. Resolution, absolute stereochemistry, and enantioselectivity of (S)-(+)- and (R)-(-)-dihydromuscimol. J Med Chem28:1612-7 (1985) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Gamma-aminobutyric acid receptor subunit gamma-1
Name:Gamma-aminobutyric acid receptor subunit gamma-1
Synonyms:Benzodiazepine receptors | Benzodiazepine receptors; peripheral & central | GABA receptor gamma-1 subunit | GBRG1_RAT | Gabrg1
Type:PROTEIN
Mol. Mass.:53557.84
Organism:Rattus norvegicus
Description:ChEMBL_193817
Residue:465
Sequence:
MGSGKVFLFSPSLLWSQTRGVRLIFLLLTLHLGNCIDKADDEDDEDLTMNKTWVLAPKIH
EGDITQILNSLLQGYDNKLRPDIGVRPTVIETDVYVNSIGPVDPINMEYTIDIIFAQTWF
DSRLKFNSTMKVLMLNSNMVGKIWIPDTFFRNSRKSDAHWITTPNRLLRIWSDGRVLYTL
RLTINAECYLQLHNFPMDEHSCPLEFSSYGYPKNEIEYKWKKPSVEVADPKYWRLYQFAF
VGLRNSTEISHTISGDYIIMTIFFDLSRRMGYFTIQTYIPCILTVVLSWVSFWINKDAVP
ARTSLGITTVLTMTTLSTIARKSLPKVSYVTAMDLFVSVCFIFVFAALMEYGTLHYFTSN
NKGKTTRDRKLKSKTSVSPGLHAGSTLIPMNNISMPQGEDDYGYQCLEGKDCATFFCCFE
DCRTGSWREGRIHIRIAKIDSYSRIFFPTAFALFNLVYWVGYLYL
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  Blast E-value cutoff:
BDBM24183
n/a
NameBDBM24183
Synonyms:4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic acid | Aminalon | CHEMBL96 | GABA | Gamma-Aminobutyric acid | [3H]GABA | cid_119
TypeRadiolabeled ligand
Emp. Form.C4H9NO2
Mol. Mass.103.1198
SMILESNCCCC(O)=O
Structure
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