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TargetAcetylpolyamine oxidase (APAO)
LigandBDBM50026233
Substrate/Competitorn/a
Meas. Tech.ChEBML_159843
Ki 425000±n/a nM
Citation Bey PBolkenius FNSeiler NCasara P N-2,3-Butadienyl-1,4-butanediamine derivatives: potent irreversible inactivators of mammalian polyamine oxidase. J Med Chem 28:1-2 (1985) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Acetylpolyamine oxidase (APAO)
Name:Polyamine oxidase
Synonyms:Peroxisomal N(1)-acetyl-spermine/spermidine oxidase | Polyamine oxidase
Type:Enzyme
Mol. Mass.:70274.33
Organism:Homo sapiens (Human)
Description:Q6QHF9
Residue:649
Sequence:
MESTGSVGEAPGGPRVLVVGGGIAGLGAAQRLCGHSAFPHLRVLEATARAGGRIRSERCF
GGVVEVGAHWIHGPSRGNPVFQLAAEYGLLGEKELSQENQLVETGGHVGLPSVSYASSGT
SVSLQLVAEMATLFYGLIDQTREFLHAAETPVPSVGEYLKKEIGQHVARLCGHSAFPHLR
VLEATARAGGRIRSERCFGGVVEVGAHWIHGPSRGNPVFQLAAEYGLLGEKELSQENQLV
ETGGHVGLPSVSYASSGASVSLQLVAEMATLFYGLIDQTREFLHAAETPVPSVGEYLKKE
IGQHVAGWTEDEETRKLKLAVLNSFFNLECCVSGTHSMDLVALAPFGEYTVLPGLDCTFS
KGYQGLTNCMMAALPEDTVVFEKPVKTIHWNGSFQEAAFPGETFPVSVECEDGDRFPAHH
VIVTVPLGFLREHLDTFFDPPLPAEKAEAIRKIGFGTNNKIFLEFEEPFWEPDCQLIQLV
WEDTSPLEDAAPELQDAWFRKLIGFVVLPAFASVHVLCGFIAGLESEFMETLSDEEVLLC
LTQVLRRVTGNPRLPAPKSVLRSRWHSAPYTRGSYSYVAVGSTGGDLDLLAQPLPADGAG
AQLQILFAGEATHRTFYSTTHGALLSGWREADRLLSLWAPQVQQPRPRL
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  Blast E-value cutoff:
BDBM50026233
n/a
NameBDBM50026233
Synonyms:CHEMBL292770 | N*1*-Prop-2-ynyl-butane-1,4-diamine
TypeSmall organic molecule
Emp. Form.C7H14N2
Mol. Mass.126.1995
SMILESNCCCCNCC#C
Structure
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