| Reaction Details |
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 | Report a problem with these data |
| Target | Chymotrypsin-like elastase family member 2A |
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| Ligand | BDBM50034579 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_152315 (CHEMBL758697) |
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| Ki | 0.365±n/a nM |
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| Citation |  Deadman, JJ; Elgendy, S; Goodwin, CA; Green, D; Baban, JA; Patel, G; Skordalakes, E; Chino, N; Claeson, G; Kakkar, VV Characterization of a class of peptide boronates with neutral P1 side chains as highly selective inhibitors of thrombin. J Med Chem38:1511-22 (1995) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Chymotrypsin-like elastase family member 2A |
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| Name: | Chymotrypsin-like elastase family member 2A |
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| Synonyms: | CEL2A_PIG | CELA2A | ELA2 | ELA2A | Elastase 2A | Elastase-2 | Elastase-2A | Pancreatic elastase |
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| Type: | PROTEIN |
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| Mol. Mass.: | 28705.23 |
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| Organism: | Sus scrofa |
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| Description: | ChEMBL_156951 |
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| Residue: | 269 |
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| Sequence: | MIRALLLSTLVAGALSCGLPANLPQLPRVVGGEDARPNSWPWQVSLQYDSSGQWRHTCGG
TLVDQSWVLTAAHCISSSRTYRVVLGRHSLSTNEPGSLAVKVSKLVVHQDWNSNQLSNGN
DIALLKLASPVSLTDKIQLGCLPAAGTILPNNYVCYVTGWGRLQTNGASPDILQQGQLLV
VDYATCSKPGWWGSTVKTNMICAGGDGIISSCNGDSGGPLNCQGANGQWQVHGIVSFGSS
LGCNYYHKPSVFTRVSNYIDWINSVIANN
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| BDBM50034579 |
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| n/a |
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| Name | BDBM50034579 |
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| Synonyms: | CHEMBL290577 | Peptide boronate |
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| Type | Small organic molecule |
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| Emp. Form. | C38H52BN3O6 |
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| Mol. Mass. | 657.647 |
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| SMILES | CCC(C)(C)C(NC(=O)[C@@H]1CCCN1C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)B1O[C@@H]2CC3CC(C3(C)C)[C@]2(C)O1 |
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| Structure | 
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