| Reaction Details |
|---|
 | Report a problem with these data |
| Target | 85/88 kDa calcium-independent phospholipase A2 |
|---|
| Ligand | BDBM50046268 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_156048 (CHEMBL760624) |
|---|
| IC50 | >100±n/a nM |
|---|
| Citation |  Zupan, LA; Weiss, RH; Hazen, SL; Parnas, BL; Aston, KW; Lennon, PJ; Getman, DP; Gross, RW Structural determinants of haloenol lactone-mediated suicide inhibition of canine myocardial calcium-independent phospholipase A2. J Med Chem36:95-100 (1993) [PubMed] |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| 85/88 kDa calcium-independent phospholipase A2 |
|---|
| Name: | 85/88 kDa calcium-independent phospholipase A2 |
|---|
| Synonyms: | Calcium-independent phospholipase A2 | PLA2G6 | PLPL9_HUMAN | PLPLA9 |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 89913.62 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | ChEMBL_156048 |
|---|
| Residue: | 806 |
|---|
| Sequence: | MQFFGRLVNTFSGVTNLFSNPFRVKEVAVADYTSSDRVREEGQLILFQNTPNRTWDCVLV
NPRNSQSGFRLFQLELEADALVNFHQYSSQLLPFYESSPQVLHTEVLQHLTDLIRNHPSW
SVAHLAVELGIRECFHHSRIISCANCAENEEGCTPLHLACRKGDGEILVELVQYCHTQMD
VTDYKGETVFHYAVQGDNSQVLQLLGRNAVAGLNQVNNQGLTPLHLACQLGKQEMVRVLL
LCNARCNIMGPNGYPIHSAMKFSQKGCAEMIISMDSSQIHSKDPRYGASPLHWAKNAEMA
RMLLKRGCNVNSTSSAGNTALHVAVMRNRFDCAIVLLTHGANADARGEHGNTPLHLAMSK
DNVEMIKALIVFGAEVDTPNDFGETPTFLASKIGRLVTRKAILTLLRTVGAEYCFPPIHG
VPAEQGSAAPHHPFSLERAQPPPISLNNLELQDLMHISRARKPAFILGSMRDEKRTHDHL
LCLDGGGVKGLIIIQLLIAIEKASGVATKDLFDWVAGTSTGGILALAILHSKSMAYMRGM
YFRMKDEVFRGSRPYESGPLEEFLKREFGEHTKMTDVRKPKVMLTGTLSDRQPAELHLFR
NYDAPETVREPRFNQNVNLRPPAQPSDQLVWRAARSSGAAPTYFRPNGRFLDGGLLANNP
TLDAMTEIHEYNQDLIRKGQANKVKKLSIVVSLGTGRSPQVPVTCVDVFRPSNPWELAKT
VFGAKELGKMVVDCCTDPDGRAVDRARAWCEMVGIQYFRLNPQLGTDIMLDEVSDTVLVN
ALWETEVYIYEHREEFQKLIQLLLSP
|
|
|
|---|
| BDBM50046268 |
|---|
| n/a |
|---|
| Name | BDBM50046268 |
|---|
| Synonyms: | 6-Bromomethylene-3-naphthalen-1-yl-tetrahydro-pyran-2-one | 6-[1-Bromo-meth-(E)-ylidene]-3-naphthalen-1-yl-tetrahydro-pyran-2-one | BTNP | CHEMBL6206 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C16H13BrO2 |
|---|
| Mol. Mass. | 317.177 |
|---|
| SMILES | Br\C=C1/CCC(C(=O)O1)c1cccc2ccccc12 |
|---|
| Structure | 
|
|---|
Search and Browse
