| Reaction Details |
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 | Report a problem with these data |
| Target | Platelet-activating factor receptor |
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| Ligand | BDBM50047772 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_221702 (CHEMBL823402) |
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| IC50 | 100±n/a nM |
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| Citation |  Trova, MP; Wissner, A; Carroll, ML; Kerwar, SS; Pickett, WC; Schaub, RE; Torley, LW; Kohler, CA Analogues of platelet activating factor. 8. Antagonists of PAF containing an aromatic ring linked to a pyridinium ring. J Med Chem36:580-90 (1993) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Platelet-activating factor receptor |
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| Name: | Platelet-activating factor receptor |
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| Synonyms: | PAF-R | PTAFR | PTAFR_CAVPO | Platelet activating factor receptor | Platelet-activating factor receptor |
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| Type: | Protein |
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| Mol. Mass.: | 39005.63 |
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| Organism: | Cavia porcellus |
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| Description: | n/a |
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| Residue: | 342 |
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| Sequence: | MELNSSSRVDSEFRYTLFPIVYSIIFVLGIIANGYVLWVFARLYPSKKLNEIKIFMVNLT
VADLLFLITLPLWIVYYSNQGNWFLPKFLCNLAGCLFFINTYCSVAFLGVITYNRFQAVK
YPIKTAQATTRKRGIALSLVIWVAIVAAASYFLVMDSTNVVSNKAGSGNITRCFEHYEKG
SKPVLIIHICIVLGFFIVFLLILFCNLVIIHTLLRQPVKQQRNAEVRRRALWMVCTVLAV
FVICFVPHHMVQLPWTLAELGMWPSSNHQAINDAHQVTLCLLSTNCVLDPVIYCFLTKKF
RKHLSEKLNIMRSSQKCSRVTTDTGTEMAIPINHTPVNPIKN
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| BDBM50047772 |
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| n/a |
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| Name | BDBM50047772 |
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| Synonyms: | CHEMBL349327 | Trifluoro-methanesulfonate2-{[acetyl-(3-methoxy-4-tetradecyloxy-benzoyl)-amino]-methyl}-1-propyl-pyridinium; |
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| Type | Small organic molecule |
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| Emp. Form. | C33H51N2O4 |
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| Mol. Mass. | 539.7685 |
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| SMILES | CCCCCCCCCCCCCCOc1ccc(cc1OC)C(=O)N(Cc1cccc[n+]1CCC)C(C)=O |
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| Structure | 
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