| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Retinoic acid receptor gamma |
|---|
| Ligand | BDBM50048293 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_196012 (CHEMBL798022) |
|---|
| Ki | 27±n/a nM |
|---|
| Citation |  Charpentier, B; Bernardon, JM; Eustache, J; Millois, C; Martin, B; Michel, S; Shroot, B Synthesis, structure-affinity relationships, and biological activities of ligands binding to retinoic acid receptor subtypes. J Med Chem38:4993-5006 (1996) [PubMed] |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Retinoic acid receptor gamma |
|---|
| Name: | Retinoic acid receptor gamma |
|---|
| Synonyms: | NR1B3 | Nuclear receptor subfamily 1 group B member 3 | RAR-gamma | RARG | RARG_HUMAN | Retinoic acid receptor RXR-alpha/gamma | Retinoic acid receptor gamma | Retinoid receptor |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 50345.43 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | ChEMBL_1458016 |
|---|
| Residue: | 454 |
|---|
| Sequence: | MATNKERLFAAGALGPGSGYPGAGFPFAFPGALRGSPPFEMLSPSFRGLGQPDLPKEMAS
LSVETQSTSSEEMVPSSPSPPPPPRVYKPCFVCNDKSSGYHYGVSSCEGCKGFFRRSIQK
NMVYTCHRDKNCIINKVTRNRCQYCRLQKCFEVGMSKEAVRNDRNKKKKEVKEEGSPDSY
ELSPQLEELITKVSKAHQETFPSLCQLGKYTTNSSADHRVQLDLGLWDKFSELATKCIIK
IVEFAKRLPGFTGLSIADQITLLKAACLDILMLRICTRYTPEQDTMTFSDGLTLNRTQMH
NAGFGPLTDLVFAFAGQLLPLEMDDTETGLLSAICLICGDRMDLEEPEKVDKLQEPLLEA
LRLYARRRRPSQPYMFPRMLMKITDLRGISTKGAERAITLKMEIPGPMPPLIREMLENPE
MFEDDSSQPGPHPNASSEDEVPGGQGKGGLKSPA
|
|
|
|---|
| BDBM50048293 |
|---|
| n/a |
|---|
| Name | BDBM50048293 |
|---|
| Synonyms: | 4-{(E)-2-[4-Hydroxy-3-(1-methyl-cyclohexyl)-phenyl]-propenyl}-benzoic acid | CHEMBL345022 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C23H26O3 |
|---|
| Mol. Mass. | 350.4507 |
|---|
| SMILES | C\C(=C/c1ccc(cc1)C(O)=O)c1ccc(O)c(c1)C1(C)CCCCC1 |
|---|
| Structure | 
|
|---|
Search and Browse
