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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | D(2) dopamine receptor | ||
| Ligand | BDBM50055731 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | ChEMBL_62399 (CHEMBL872888) | ||
| Ki | 28±n/a nM | ||
| Citation |  Wustrow, DJ; Smith, WJ; Corbin, AE; Davis, MD; Georgic, LM; Pugsley, TA; Whetzel, SZ; Heffner, TG; Wise, LD 3-[[(4-Aryl-1-piperazinyl)alkyl]cyclohexyl]-1H-indoles as dopamine D2 partial agonists and autoreceptor agonists. J Med Chem40:250-9 (1997) [PubMed] Article | ||
| More Info.: | Get all data from this article, Assay Method | ||
| D(2) dopamine receptor | |||
| Name: | D(2) dopamine receptor | ||
| Synonyms: | DOPAMINE D2 | DOPAMINE D2 Long | DOPAMINE D2 Short | DRD2_RAT | Dopamine D2 receptor | Dopamine2-like | Drd2 | ||
| Type: | G Protein-Coupled Receptor (GPCR) | ||
| Mol. Mass.: | 50931.60 | ||
| Organism: | Rattus norvegicus (rat) | ||
| Description: | P61169 | ||
| Residue: | 444 | ||
| Sequence: |
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| BDBM50055731 | |||
| n/a | |||
| Name | BDBM50055731 | ||
| Synonyms: | 3-{4-[2-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-ethyl]-cyclohexyl}-1H-indole | CHEMBL87003 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C27H32N2 | ||
| Mol. Mass. | 384.5564 | ||
| SMILES | C(CN1CCC(=CC1)c1ccccc1)[C@H]1CC[C@H](CC1)c1c[nH]c2ccccc12 |wU:17.22,14.15,c:5,(13.37,-6.33,;14.69,-7.1,;16.03,-6.36,;17.35,-7.1,;18.69,-6.33,;18.67,-4.79,;17.32,-4.02,;16.01,-4.82,;20,-4.02,;21.33,-4.79,;22.66,-4.02,;22.64,-2.48,;21.32,-1.71,;19.98,-2.48,;12.03,-7.1,;12.02,-8.63,;10.71,-9.37,;9.37,-8.6,;9.37,-7.1,;10.71,-6.33,;8.09,-9.47,;8.02,-11.01,;6.54,-11.42,;5.68,-10.14,;4.15,-9.92,;3.6,-8.47,;4.58,-7.26,;6.09,-7.51,;6.65,-8.92,)| | ||
| Structure | 
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