| Reaction Details |
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 | Report a problem with these data |
| Target | Sigma non-opioid intracellular receptor 1 |
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| Ligand | BDBM50065143 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_200969 (CHEMBL802057) |
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| Ki | 3.11±n/a nM |
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| Citation |  John, CS; Lim, BB; Vilner, BJ; Geyer, BC; Bowen, WD Substituted halogenated arylsulfonamides: a new class of sigma receptor binding tumor imaging agents. J Med Chem41:2445-50 (1998) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Sigma non-opioid intracellular receptor 1 |
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| Name: | Sigma non-opioid intracellular receptor 1 |
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| Synonyms: | Aging-associated gene 8 protein | OPRS1 | SGMR1_HUMAN | SIG-1R | SIGMAR1 | SR-BP | SR31747-binding protein | SRBP | Sigma 1-type opioid receptor | Sigma opioid receptor | Sigma1R | hSigmaR1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 25124.85 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Q99720 |
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| Residue: | 223 |
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| Sequence: | MQWAVGRRWAWAALLLAVAAVLTQVVWLWLGTQSFVFQREEIAQLARQYAGLDHELAFSR
LIVELRRLHPGHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSRGHSGRY
WAEISDTIISGTFHQWREGTTKSEVFYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPS
TLAFALADTVFSTQDFLTLFYTLRSYARGLRLELTTYLFGQDP
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| BDBM50065143 |
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| n/a |
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| Name | BDBM50065143 |
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| Synonyms: | CHEMBL83448 | N-(2-Azepan-1-yl-ethyl)-3-iodo-4-methoxy-N-methyl-benzenesulfonamide |
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| Type | Small organic molecule |
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| Emp. Form. | C16H25IN2O3S |
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| Mol. Mass. | 452.351 |
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| SMILES | COc1ccc(cc1I)S(=O)(=O)N(C)CCN1CCCCCC1 |
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| Structure | 
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