| Reaction Details |
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 | Report a problem with these data |
| Target | Somatostatin receptor type 2 |
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| Ligand | BDBM50065451 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_200363 (CHEMBL807430) |
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| Kd | 407±n/a nM |
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| Citation |  Tran, TA; Mattern, RH; Afargan, M; Amitay, O; Ziv, O; Morgan, BA; Taylor, JE; Hoyer, D; Goodman, M Design, synthesis, and biological activities of potent and selective somatostatin analogues incorporating novel peptoid residues. J Med Chem41:2679-85 (1998) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Somatostatin receptor type 2 |
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| Name: | Somatostatin receptor type 2 |
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| Synonyms: | SOMATOSTATIN SST2 | SRIF-1 | SS-2-R | SS2-R | SS2R | SSR2_HUMAN | SSTR2 | Somatostatin receptor type 2 (SSTR2) |
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| Type: | Enzyme |
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| Mol. Mass.: | 41344.94 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P30874 |
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| Residue: | 369 |
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| Sequence: | MDMADEPLNGSHTWLSIPFDLNGSVVSTNTSNQTEPYYDLTSNAVLTFIYFVVCIIGLCG
NTLVIYVILRYAKMKTITNIYILNLAIADELFMLGLPFLAMQVALVHWPFGKAICRVVMT
VDGINQFTSIFCLTVMSIDRYLAVVHPIKSAKWRRPRTAKMITMAVWGVSLLVILPIMIY
AGLRSNQWGRSSCTINWPGESGAWYTGFIIYTFILGFLVPLTIICLCYLFIIIKVKSSGI
RVGSSKRKKSEKKVTRMVSIVVAVFIFCWLPFYIFNVSSVSMAISPTPALKGMFDFVVVL
TYANSCANPILYAFLSDNFKKSFQNVLCLVKVSGTDDGERSDSKQDKSRLNETTETQRTL
LNGDLQTSI
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| BDBM50065451 |
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| n/a |
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| Name | BDBM50065451 |
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| Synonyms: | 2-Amino-N-{4-[(2S,5S,8S,14S,17R)-8,14-dibenzyl-5-((R)-1-hydroxy-ethyl)-17-(1H-indol-3-ylmethyl)-3,6,9,12,15,18-hexaoxo-10-((R)-1-phenyl-ethyl)-1,4,7,10,13,16hexaaza-cyclooctadec-2-yl]-butyl}-3-phenyl-propionamide | CHEMBL2370167 |
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| Type | Small organic molecule |
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| Emp. Form. | C58H67N9O8 |
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| Mol. Mass. | 1018.2081 |
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| SMILES | [H][C@]1(NC(=O)[C@H](CCCCNC(=O)[C@@H](N)Cc2ccccc2)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC(=O)CN([C@H](C)c2ccccc2)C(=O)[C@H](Cc2ccccc2)NC1=O)[C@@H](C)O |
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| Structure | 
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