Reaction Details |
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Target | Mu-type opioid receptor |
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Ligand | BDBM50067447 |
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Substrate/Competitor | n/a |
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Meas. Tech. | ChEMBL_145301 (CHEMBL752836) |
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Ki | 0.34±n/a nM |
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Citation | Thomas, JB; Zheng, X; Mascarella, SW; Rothman, RB; Dersch, CM; Partilla, JS; Flippen-Anderson, JL; George, CF; Cantrell, BE; Zimmerman, DM; Carroll, FI N-Substituted 9beta-methyl-5-(3-hydroxyphenyl)morphans are opioid receptor pure antagonists. J Med Chem41:4143-9 (1998) [PubMed] Article |
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More Info.: | Get all data from this article, Assay Method |
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Mu-type opioid receptor |
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Name: | Mu-type opioid receptor |
Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 11165.58 |
Organism: | GUINEA PIG |
Description: | P97266 |
Residue: | 98 |
Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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BDBM50067447 |
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n/a |
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Name | BDBM50067447 |
Synonyms: | 3-((R)-9-Methyl-2-phenethyl-2-aza-bicyclo[3.3.1]non-5-yl)-phenol | CHEMBL334898 |
Type | Small organic molecule |
Emp. Form. | C23H29NO |
Mol. Mass. | 335.4825 |
SMILES | C[C@H]1C2CCCC1(CCN2CCc1ccccc1)c1cccc(O)c1 |
Structure |
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