| Reaction Details |
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 | Report a problem with these data |
| Target | Tryptase gamma |
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| Ligand | BDBM50067522 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_210825 (CHEMBL811854) |
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| IC50 | 29000±n/a nM |
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| Citation |  Gabriel, B; Stubbs, MT; Bergner, A; Hauptmann, J; Bode, W; Stürzebecher, J; Moroder, L Design of benzamidine-type inhibitors of factor Xa. J Med Chem41:4240-50 (1998) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Tryptase gamma |
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| Name: | Tryptase gamma |
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| Synonyms: | PRSS31 | Serine protease 31 | TMT | TPSG1 | TRYG1_HUMAN | Transmembrane tryptase | Tryptase | Tryptase gamma | Tryptase gamma heavy chain | Tryptase gamma light chain |
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| Type: | PROTEIN |
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| Mol. Mass.: | 33817.52 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_210833 |
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| Residue: | 321 |
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| Sequence: | MALGACGLLLLLAVPGVSLRTLQPGCGRPQVSDAGGRIVGGHAAPAGAWPWQASLRLRRM
HVCGGSLLSPQWVLTAAHCFSGSLNSSDYQVHLGELEITLSPHFSTVRQIILHSSPSGQP
GTSGDIALVELSVPVTLSSRILPVCLPEASDDFCPGIRCWVTGWGYTREGEPLPPPYSLR
EVKVSVVDTETCRRDYPGPGGSILQPDMLCARGPGDACQDDSGGPLVCQVNGAWVQAGTV
SWGEGCGRPNRPGVYTRVPAYVNWIRRHITASGGSESGYPRLPLLAGLFLPGLFLLLVSC
VLLAKCLLHPSADGTPFPAPD
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| BDBM50067522 |
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| n/a |
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| Name | BDBM50067522 |
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| Synonyms: | 2-[2-(4-Carbamimidoyl-benzenesulfonylamino)-acetylamino]-3-(4-carbamimidoyl-phenyl)-propionic acid ethyl ester | CHEMBL135815 |
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| Type | Small organic molecule |
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| Emp. Form. | C21H26N6O5S |
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| Mol. Mass. | 474.533 |
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| SMILES | CCOC(=O)C(Cc1ccc(cc1)C(N)=N)NC(=O)CNS(=O)(=O)c1ccc(cc1)C(N)=N |
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| Structure | 
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