| Reaction Details |
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 | Report a problem with these data |
| Target | Potassium voltage-gated channel subfamily A member 2 |
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| Ligand | BDBM50067878 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_92807 (CHEMBL703985) |
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| Kd | 590000±n/a nM |
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| Citation |  Wulff, H; Rauer, H; Düring, T; Hanselmann, C; Ruff, K; Wrisch, A; Grissmer, S; Hänsel, W Alkoxypsoralens, novel nonpeptide blockers of Shaker-type K+ channels: synthesis and photoreactivity. J Med Chem41:4542-9 (1998) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Potassium voltage-gated channel subfamily A member 2 |
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| Name: | Potassium voltage-gated channel subfamily A member 2 |
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| Synonyms: | HBK5 | HUKIV | KCNA2 | KCNA2_HUMAN | NGK1 | Potassium voltage-gated channel subfamily A member 2 | Voltage-gated potassium channel | Voltage-gated potassium channel subunit Kv1.2 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 56695.97 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_334898 |
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| Residue: | 499 |
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| Sequence: | MTVATGDPADEAAALPGHPQDTYDPEADHECCERVVINISGLRFETQLKTLAQFPETLLG
DPKKRMRYFDPLRNEYFFDRNRPSFDAILYYYQSGGRLRRPVNVPLDIFSEEIRFYELGE
EAMEMFREDEGYIKEEERPLPENEFQRQVWLLFEYPESSGPARIIAIVSVMVILISIVSF
CLETLPIFRDENEDMHGSGVTFHTYSNSTIGYQQSTSFTDPFFIVETLCIIWFSFEFLVR
FFACPSKAGFFTNIMNIIDIVAIIPYFITLGTELAEKPEDAQQGQQAMSLAILRVIRLVR
VFRIFKLSRHSKGLQILGQTLKASMRELGLLIFFLFIGVILFSSAVYFAEADERESQFPS
IPDAFWWAVVSMTTVGYGDMVPTTIGGKIVGSLCAIAGVLTIALPVPVIVSNFNYFYHRE
TEGEEQAQYLQVTSCPKIPSSPDLKKSRSASTISKSDYMEIQEGVNNSNEDFREENLKTA
NCTLANTNYVNITKMLTDV
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| BDBM50067878 |
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| n/a |
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| Name | BDBM50067878 |
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| Synonyms: | 9-Methoxy-furo[3',2':4,5]benzo[1,2-b][1,4]oxazin-3-one | CHEMBL141623 |
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| Type | Small organic molecule |
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| Emp. Form. | C11H7NO4 |
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| Mol. Mass. | 217.1776 |
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| SMILES | COc1c2ccoc2cc2oc(=O)cnc12 |
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| Structure | 
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