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TargetPotassium voltage-gated channel subfamily A member 5
LigandBDBM50067880
Substrate/Competitorn/a
Meas. Tech.ChEMBL_92809 (CHEMBL702905)
Kd 177000±n/a nM
Citation Wulff, H; Rauer, H; Düring, T; Hanselmann, C; Ruff, K; Wrisch, A; Grissmer, S; Hänsel, W Alkoxypsoralens, novel nonpeptide blockers of Shaker-type K+ channels: synthesis and photoreactivity. J Med Chem41:4542-9 (1998) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Potassium voltage-gated channel subfamily A member 5
Name:Potassium voltage-gated channel subfamily A member 5
Synonyms:HK2 | HPCN1 | KCNA5 | KCNA5_HUMAN | Potassium voltage-gated channel subfamily A member 5 | Voltage-gated potassium channel | Voltage-gated potassium channel subunit Kv1.5
Type:Enzyme
Mol. Mass.:67222.47
Organism:Homo sapiens (Human)
Description:P22460
Residue:613
Sequence:
MEIALVPLENGGAMTVRGGDEARAGCGQATGGELQCPPTAGLSDGPKEPAPKGRGAQRDA
DSGVRPLPPLPDPGVRPLPPLPEELPRPRRPPPEDEEEEGDPGLGTVEDQALGTASLHHQ
RVHINISGLRFETQLGTLAQFPNTLLGDPAKRLRYFDPLRNEYFFDRNRPSFDGILYYYQ
SGGRLRRPVNVSLDVFADEIRFYQLGDEAMERFREDEGFIKEEEKPLPRNEFQRQVWLIF
EYPESSGSARAIAIVSVLVILISIITFCLETLPEFRDERELLRHPPAPHQPPAPAPGANG
SGVMAPPSGPTVAPLLPRTLADPFFIVETTCVIWFTFELLVRFFACPSKAGFSRNIMNII
DVVAIFPYFITLGTELAEQQPGGGGGGQNGQQAMSLAILRVIRLVRVFRIFKLSRHSKGL
QILGKTLQASMRELGLLIFFLFIGVILFSSAVYFAEADNQGTHFSSIPDAFWWAVVTMTT
VGYGDMRPITVGGKIVGSLCAIAGVLTIALPVPVIVSNFNYFYHRETDHEEPAVLKEEQG
TQSQGPGLDRGVQRKVSGSRGSFCKAGGTLENADSARRGSCPLEKCNVKAKSNVDLRRSL
YALCLDTSRETDL
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50067880
n/a
NameBDBM50067880
Synonyms:4-methoxy-7H-furo[3,2-g][1]benzopyran-7-one | 4-methoxy-7H-furo[3,2-g]chromen-7-one | 5-methoxypsoralen | 5-methoxypsoralene | Bergaptene | CHEMBL24171 | Heraclin | Majudin
TypeSmall organic molecule
Emp. Form.C12H8O4
Mol. Mass.216.1895
SMILESCOc1c2ccoc2cc2oc(=O)ccc12
Structure
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