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TargetDelta-type opioid receptor
LigandBDBM50068136
Substrate/Competitorn/a
Meas. Tech.ChEMBL_124881 (CHEMBL731341)
EC50 174±n/a nM
Citation Liao, SAlfaro-Lopez, JShenderovich, MDHosohata, KLin, JLi, XStropova, DDavis, PJernigan, KAPorreca, FYamamura, HIHruby, VJ De novo design, synthesis, and biological activities of high-affinity and selective non-peptide agonists of the delta-opioid receptor. J Med Chem41:4767-76 (1998) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Delta-type opioid receptor
Name:Delta-type opioid receptor
Synonyms:DOR-1 | K56 | MSL-2 | OPIATE Delta | OPRD_MOUSE | Opioid receptors; mu and delta | Oprd1
Type:Enzyme Catalytic Domain
Mol. Mass.:40577.25
Organism:MOUSE
Description:P32300
Residue:372
Sequence:
MELVPSARAELQSSPLVNLSDAFPSAFPSAGANASGSPGARSASSLALAIAITALYSAVC
AVGLLGNVLVMFGIVRYTKLKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELL
CKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVG
VPIMVMAVTQPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRL
RSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDINRRDPLVVAAL
HLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRTPCGRQEPGSLRRPRQATTRERVTAC
TPSDGPGGGAAA
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  Blast E-value cutoff:
BDBM50068136
n/a
NameBDBM50068136
Synonyms:3-[(4-Benzyl-piperazin-1-yl)-phenyl-methyl]-phenol | CHEMBL356587
TypeSmall organic molecule
Emp. Form.C24H26N2O
Mol. Mass.358.476
SMILESOc1cccc(c1)C(N1CCN(Cc2ccccc2)CC1)c1ccccc1
Structure
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