| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50070946 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_138741 |
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| Ki | 1015±n/a nM |
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| Citation |  Tsai, YC; Liou, JP; Liao, R; Cheng, CY; Tao, PL C-alkylated spiro[benzofuran-3(2H),4'-1'-methyl-piperidine-7-ols] as potent opioids: a conformation-activity study. Bioorg Med Chem Lett8:1813-8 (1999) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 11165.58 |
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| Organism: | GUINEA PIG |
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| Description: | P97266 |
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| Residue: | 98 |
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| Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
|
|
|
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| BDBM50070946 |
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| n/a |
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| Name | BDBM50070946 |
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| Synonyms: | 1',3'-dimethylspiro[2,3-dihydrobenzo[b]furan-3,4'-(hexahydropyridine)]-7-ol | CHEMBL300689 |
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| Type | Small organic molecule |
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| Emp. Form. | C14H19NO2 |
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| Mol. Mass. | 233.3062 |
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| SMILES | CC1CN(C)CCC11COc2c1cccc2O |
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| Structure | 
|
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