| Reaction Details |
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 | Report a problem with these data |
| Target | Histamine H3 receptor |
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| Ligand | BDBM50071488 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_85851 |
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| Ki | 38±n/a nM |
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| Citation |  Aslanian, R; Brown, JE; Shih, NY; wa Mutahi, M; Green, MJ; She, S; Del Prado, M; West, R; Hey, J 4-[(1H-imidazol-4-yl) methyl] benzamidines and benzylamidines: novel antagonists of the histamine H3 receptor. Bioorg Med Chem Lett8:2263-8 (1999) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Histamine H3 receptor |
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| Name: | Histamine H3 receptor |
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| Synonyms: | HISTAMINE H3 | HRH3 | HRH3_CAVPO | Histamine H3 receptor |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 48753.61 |
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| Organism: | GUINEA PIG |
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| Description: | HISTAMINE H3 HRH3 GUINEA PIG::Q9JI35 |
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| Residue: | 445 |
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| Sequence: | MERAPPDGLMNASGALAGEAAAAAGGARTFSAAWTAVLAALMALLIVATVLGNALVMLAF
VADSSLRTQNNFFLLNLAISDFLVGVFCIPLYVPYVLTGRWTFGRGLCKLWLVVDYLLCT
SSVFNIVLISYDRFLSVTRAVSYRAQQGDTRRAVRKMVLVWVLAFLLYGPAILSWEYLSG
GSSIPEGHCYAEFFYNWYFLITASTLEFFTPFLSVTFFNLSIYLNIQRRTRLRLDGGARE
AGPDPLPEAQSSPPQPPPGCWGCWPKGQGESMPLHRYGVGEAGPGAEAGEAALGGGSGAA
ASPTSSSGSSSRGTERPRSLKRGSKPSASSASLEKRMKMVSQSITQRFRLSRDKKVAKSL
AIIVSIFGLCWAPYTLLMIIRAACHGHCVPDYWYETSFWLLWANSAVNPVLYPLCHYSFR
RAFTKLLCPQKLKVQPHSSLEHCWK
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| BDBM50071488 |
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| n/a |
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| Name | BDBM50071488 |
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| Synonyms: | 4-(1H-Imidazol-4-ylmethyl)-benzamidine | CHEMBL73605 |
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| Type | Small organic molecule |
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| Emp. Form. | C11H12N4 |
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| Mol. Mass. | 200.2398 |
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| SMILES | NC(=N)c1ccc(Cc2cnc[nH]2)cc1 |
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| Structure | 
|
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