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TargetGag-Pol polyprotein [489-587]
LigandBDBM50073267
Substrate/Competitorn/a
Meas. Tech.ChEBML_157700
Ki 1.2±n/a nM
Citation Randad, RSLubkowska, LEissenstat, MAGulnik, SVYu, BBhat, TNClanton, DJHouse, TStinson, SFErickson, JW Unsymmetric nonpeptidic HIV protease inhibitors containing anthranilamide as a P2' ligand. Bioorg Med Chem Lett8:3537-42 (1999) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Gag-Pol polyprotein [489-587]
Name:Gag-Pol polyprotein [489-587]
Synonyms:Human immunodeficiency virus type 1 protease | POL_HV1H2 | Pol polyprotein | gag-pol
Type:Enzyme Subunit
Mol. Mass.:10781.16
Organism:Human immunodeficiency virus type 1
Description:P04585[489-587]
Residue:99
Sequence:
PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYD
QILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF
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  Blast E-value cutoff:
BDBM50073267
n/a
NameBDBM50073267
Synonyms:(2-{(1S,3S,4S)-1-Benzyl-3-hydroxy-4-[(isoxazole-5-carbonyl)-amino]-5-phenyl-pentylcarbamoyl}-phenyl)-carbamic acid pyridin-2-ylmethyl ester | CHEMBL333337
TypeSmall organic molecule
Emp. Form.C36H35N5O6
Mol. Mass.633.693
SMILESO[C@@H](C[C@H](Cc1ccccc1)NC(=O)c1ccccc1NC(=O)OCc1ccccn1)[C@H](Cc1ccccc1)NC(=O)c1ccno1
Structure
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