| Reaction Details |
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 | Report a problem with these data |
| Target | Chymotrypsin-like elastase family member 2A |
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| Ligand | BDBM50075111 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_158076 |
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| IC50 | 180±n/a nM |
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| Citation |  Iijima, K; Katada, J; Hayashi, Y Symmetrical anhydride-type serine protease inhibitors: structure-activity relationship studies of human chymase inhibitors. Bioorg Med Chem Lett9:413-8 (1999) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Chymotrypsin-like elastase family member 2A |
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| Name: | Chymotrypsin-like elastase family member 2A |
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| Synonyms: | CEL2A_PIG | CELA2A | ELA2 | ELA2A | Elastase 2A | Elastase-2 | Elastase-2A | Pancreatic elastase |
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| Type: | PROTEIN |
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| Mol. Mass.: | 28705.23 |
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| Organism: | Sus scrofa |
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| Description: | ChEMBL_156951 |
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| Residue: | 269 |
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| Sequence: | MIRALLLSTLVAGALSCGLPANLPQLPRVVGGEDARPNSWPWQVSLQYDSSGQWRHTCGG
TLVDQSWVLTAAHCISSSRTYRVVLGRHSLSTNEPGSLAVKVSKLVVHQDWNSNQLSNGN
DIALLKLASPVSLTDKIQLGCLPAAGTILPNNYVCYVTGWGRLQTNGASPDILQQGQLLV
VDYATCSKPGWWGSTVKTNMICAGGDGIISSCNGDSGGPLNCQGANGQWQVHGIVSFGSS
LGCNYYHKPSVFTRVSNYIDWINSVIANN
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| BDBM50075111 |
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| n/a |
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| Name | BDBM50075111 |
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| Synonyms: | 2-(4-cyanophenylcarboxamido)-2-cyclohex-3-enyl-1,1-dimethylpropanoic anhydride | CHEMBL134024 |
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| Type | Small organic molecule |
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| Emp. Form. | C38H42N4O5 |
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| Mol. Mass. | 634.7639 |
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| SMILES | CC(C)(C(NC(=O)c1ccc(cc1)C#N)C1CCC=CC1)C(=O)OC(=O)C(C)(C)C(NC(=O)c1ccc(cc1)C#N)C1CCC=CC1 |c:19,47| |
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| Structure | 
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