| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Beta-1 adrenergic receptor |
|---|
| Ligand | BDBM50077647 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEBML_37401 |
|---|
| Kd | 120±n/a nM |
|---|
| Citation |  Suzuki, H; Shindo, K; Ueno, A; Miura, T; Takei, M; Sakakibara, M; Fukamachi, H; Tanaka, J; Higa, T S1319: a novel beta2-andrenoceptor agonist from a marine sponge Dysidea sp. Bioorg Med Chem Lett9:1361-4 (1999) [PubMed] |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Beta-1 adrenergic receptor |
|---|
| Name: | Beta-1 adrenergic receptor |
|---|
| Synonyms: | ADRB1 | ADRB1R | ADRB1_HUMAN | B1AR | Beta-1 adrenoceptor | adrenergic Beta1 |
|---|
| Type: | G Protein-Coupled Receptor (GPCR) |
|---|
| Mol. Mass.: | 51338.40 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P08588 |
|---|
| Residue: | 477 |
|---|
| Sequence: | MGAGVLVLGASEPGNLSSAAPLPDGAATAARLLVPASPPASLLPPASESPEPLSQQWTAG
MGLLMALIVLLIVAGNVLVIVAIAKTPRLQTLTNLFIMSLASADLVMGLLVVPFGATIVV
WGRWEYGSFFCELWTSVDVLCVTASIETLCVIALDRYLAITSPFRYQSLLTRARARGLVC
TVWAISALVSFLPILMHWWRAESDEARRCYNDPKCCDFVTNRAYAIASSVVSFYVPLCIM
AFVYLRVFREAQKQVKKIDSCERRFLGGPARPPSPSPSPVPAPAPPPGPPRPAAAAATAP
LANGRAGKRRPSRLVALREQKALKTLGIIMGVFTLCWLPFFLANVVKAFHRELVPDRLFV
FFNWLGYANSAFNPIIYCRSPDFRKAFQRLLCCARRAARRRHATHGDRPRASGCLARPGP
PPSPGAASDDDDDDVVGATPPARLLEPWAGCNGGAAADSDSSLDEPCRPGFASESKV
|
|
|
|---|
| BDBM50077647 |
|---|
| n/a |
|---|
| Name | BDBM50077647 |
|---|
| Synonyms: | 4-Hydroxy-7-(1-hydroxy-2-methylamino-ethyl)-3H-benzothiazol-2-one | 4-hydroxy-7-(1-hydroxy-2-(methylamino)ethyl)benzo[d]thiazol-2(3H)-one | CHEMBL29141 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C10H12N2O3S |
|---|
| Mol. Mass. | 240.279 |
|---|
| SMILES | CNCC(O)c1ccc(O)c2[nH]c(=O)sc12 |
|---|
| Structure | 
|
|---|
Search and Browse
