| Reaction Details |
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 | Report a problem with these data |
| Target | Kallikrein-1 |
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| Ligand | BDBM50079380 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_92369 (CHEMBL701583) |
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| Ki | >10000000±n/a nM |
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| Citation |  Sanders, TC; Seto, CT 4-Heterocyclohexanone-based inhibitors of the serine protease plasmin. J Med Chem42:2969-76 (1999) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Kallikrein-1 |
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| Name: | Kallikrein-1 |
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| Synonyms: | KLK1 | KLK1_HUMAN | Kallikrein 1 | Kallikrein-1 | Kidney/pancreas/salivary gland kallikrein | Tissue kallikrein |
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| Type: | Enzyme |
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| Mol. Mass.: | 28874.69 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P06870 |
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| Residue: | 262 |
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| Sequence: | MWFLVLCLALSLGGTGAAPPIQSRIVGGWECEQHSQPWQAALYHFSTFQCGGILVHRQWV
LTAAHCISDNYQLWLGRHNLFDDENTAQFVHVSESFPHPGFNMSLLENHTRQADEDYSHD
LMLLRLTEPADTITDAVKVVELPTEEPEVGSTCLASGWGSIEPENFSFPDDLQCVDLKIL
PNDECKKAHVQKVTDFMLCVGHLEGGKDTCVGDSGGPLMCDGVLQGVTSWGYVPCGTPNK
PSVAVRVLSYVKWIEDTIAENS
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| BDBM50079380 |
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| n/a |
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| Name | BDBM50079380 |
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| Synonyms: | 3-[Bis-(6-amino-hexyl)-amino]-tetrahydro-thiopyran-4-one | CHEMBL318854 |
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| Type | Small organic molecule |
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| Emp. Form. | C17H35N3OS |
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| Mol. Mass. | 329.544 |
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| SMILES | NCCCCCCN(CCCCCCN)C1CSCCC1=O |
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| Structure | 
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