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TargetH2-K region expressed gene 2, rat orthologue
LigandBDBM50079848
Substrate/Competitorn/a
Meas. Tech.ChEMBL_103873 (CHEMBL712990)
IC50 100±n/a nM
Citation Jones, ABActon, JJAdams, ADYuen, WNichols, EASchwartz, CDWicker, LSHermes, JD Tetrapeptide derived inhibitors of complexation of a class II MHC: fully unnatural ligands. Bioorg Med Chem Lett9:2115-8 (1999) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
H2-K region expressed gene 2, rat orthologue
Name:H2-K region expressed gene 2, rat orthologue
Synonyms:MHC class II | MHC class II region expressed gene KE2, isoform CRA_a
Type:PROTEIN
Mol. Mass.:14499.39
Organism:Rattus norvegicus
Description:ChEMBL_10342
Residue:127
Sequence:
MAELIQKKLQGEVEKYQQLQKDLSKSMSGRQKLEAQLTENNIVKEELALLDGSNVVFKLL
GPVLVKQELGEARATVGKRLDYITAEIKRYESQLRDLERQSEQQRETLAQLQQEFQRAQN
AKAPGKA
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  Blast E-value cutoff:
BDBM50079848
n/a
NameBDBM50079848
Synonyms:(S)-2-(3-Cyclohexyl-propylamino)-2-methyl-pentanoic acid [(S)-1-((S)-1-carbamoyl-3-methyl-butylcarbamoyl)-butyl]-amide | CHEMBL67080
TypeSmall organic molecule
Emp. Form.C26H50N4O3
Mol. Mass.466.7002
SMILESCCC[C@H](NC(=O)[C@](C)(CCC)NCCCC1CCCCC1)C(=O)N[C@@H](CC(C)C)C(N)=O
Structure
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