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TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 2
LigandBDBM50080528
Substrate/Competitorn/a
Meas. Tech.ChEMBL_153000
Ki 187000±n/a nM
Citation Christner CWyrwa RMarsch SKüllertz GThiericke RGrabley SSchumann DFischer G Synthesis and cytotoxic evaluation of cycloheximide derivatives as potential inhibitors of FKBP12 with neuroregenerative properties. J Med Chem 42:3615-22 (1999) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 2
Name:Peptidyl-prolyl cis-trans isomerase NIMA-interacting 2
Synonyms:PPIase Pin4 | Par14 | Parvulin 14 | Peptidyl-prolyl cis-trans isomerase NIMA-interacting 4 | Peptidyl-prolyl cis/trans isomerase EPVH | Rotamase Pin4 | hPar14
Type:PROTEIN
Mol. Mass.:13820.38
Organism:Homo sapiens (Human)
Description:ChEMBL_1502606
Residue:131
Sequence:
MPPKGKSGSGKAGKGGAASGSDSADKKAQGPKGGGNAVKVRHILCEKHGKIMEAMEKLKS
GMRFNEVAAQYSEDKARQGGDLGWMTRGSMVGPFQEAAFALPVSGMDKPVFTDPPVKTKF
GYHIIMVEGRK
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  Blast E-value cutoff:
BDBM50080528
n/a
NameBDBM50080528
Synonyms:3-((R)-2-((1S,3S,5S)-3,5-dimethyl-2-oxocyclohexyl)-2-hydroxyethyl)glutarimide | 4-{(2R)-2-[(1S,3S,5S)-3,5-dimethyl-2-oxocyclohexyl]-2-hydroxyethyl}piperidine-2,6-dione | CHEMBL123292 | Cycloheximid | Zykloheximid | cid_6197 | cycloheximide
TypeSmall organic molecule
Emp. Form.C15H23NO4
Mol. Mass.281.3474
SMILESC[C@H]1C[C@H](C)C(=O)[C@@H](C1)[C@H](O)CC1CC(=O)NC(=O)C1 |r|
Structure
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